SCHEMBL4357095

SCHEMBL4357095

CCn1cnc2c(=O)nc(Cl)n(-c3ccc(F)cc3)c21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 2/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
RXFP1 Q9HBX9 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PTGS2 P35354 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CDK1 P06493 3/20 0.35
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2233449 0.81 MAT2A (0.42) MAT2ANPC1RAB9ASMN1; SMN2LMNA
SCHEMBL4778102 0.80 MAPK1 (0.36) NPC1RAB9ASMN1; SMN2TSHRPDE4A
SCHEMBL4772467 0.79 MAT2A (0.40) MAT2ANPC1RAB9ASMN1; SMN2LMNA
SCHEMBL4776782 0.78 CDK1 (0.33) MAT2ANPC1RAB9ASMN1; SMN2LMNA
SCHEMBL5769775 0.77 NPSR1 (0.37) MAT2ANPC1RAB9ASMN1; SMN2LMNA
SCHEMBL4768907 0.77 SMN1; SMN2 (0.34) MAT2ANPC1RAB9ASMN1; SMN2LMNA
SCHEMBL4260069 0.76 AXL (0.36) CYP1A2KDM4EALDH1A1GAAL3MBTL1
SCHEMBL4284448 0.76 NPC1 (0.34) NPC1RAB9ASMN1; SMN2LMNAHPGD
SCHEMBL4256906 0.76 BRD4 (0.40) CYP2C19
SCHEMBL4768956 0.76 SCN9A (0.34) NPC1RAB9ASMN1; SMN2LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094704-A2 CIS-CYCLOHEXYL SUBSTITUTED PYRIMIDINONE DERIVATIVES Neurogen Corporation (US) 2009-09-02 EP disclosed
WO-2008066664-A2 CIS-CYCLOHEXYL SUBSTITUTED PYRIMIDINONE DERIVATIVES NEUROGEN CORPORATION (US) 2008-06-05 WO disclosed