SCHEMBL435715

SCHEMBL435715

O=C(NO)C1CCc2ccc(CCNc3cccc(Cl)c3)cc2C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.40
MAPT P10636 3/20 0.40
KMT2A Q03164 3/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
HDAC6 Q9UBN7 2/20 0.39
HDAC1 Q13547 2/20 0.39
TAAR1 Q96RJ0 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC2 Q92769 1/20 0.39
GLA P06280 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HDAC8 Q9BY41 2/20 0.39
MAOB P27338 1/20 0.39
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL345656 0.82 MAOB (0.43) MEN1MAPTKMT2ALMNACYP1A2
SCHEMBL346576 0.78 GRIN2B (0.44) HDAC1
SCHEMBL346051 0.77 CA1 (0.47) KMT2AHDAC6HDAC8MAOB
SCHEMBL435714 0.76 S1PR1 (0.39) MEN1MAPTKMT2ALMNACYP1A2
SCHEMBL10197649 0.74 ADRB3 (0.49) HDAC6HDAC8
SCHEMBL435688 0.70 ADRB3 (0.47) HDAC6HDAC1HDAC2HDAC8
SCHEMBL436766 0.70 NR1H2 (0.39) ALDH1A1
SCHEMBL346158 0.70 HDAC1 (0.44) MAPTHDAC1
SCHEMBL346594 0.70 FFAR1 (0.48)
SCHEMBL460177 0.70 FAAH (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012320-A1 SUBSTITUTED HYDROXAMIC ACIDS AND USES THEREOF MILLENIUM PHARMACEUTICALS, INC. (US) 2012-01-26 WO disclosed