SCHEMBL4357530

SCHEMBL4357530

CC(C)NC(=O)N(S)c1ccc(O)c([N+](=O)[O-])c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
MAPK1 P28482 2/20 0.42
HPGD P15428 2/20 0.42
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
GPR35 Q9HC97 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAPT P10636 4/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ALDH5A1 P51649 1/20 0.39
ABAT P80404 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
KDM4E B2RXH2 2/20 0.38
USP2 O75604 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4353654 0.78 MAPT (0.49) ALDH1A1MAPK1HPGDTP53TSHR
SCHEMBL4343483 0.78 ESR1 (0.39) ALDH1A1HSD17B10KDM4ELMNA
SCHEMBL4357469 0.78 MAPK1 (0.38) ALDH1A1MAPK1TSHRSMN1; SMN2HSD17B10
SCHEMBL4345611 0.78 MAPT (0.42) ALDH1A1MAPK1HPGDTP53TSHR
SCHEMBL4356327 0.77 TRPV1 (0.45) ALDH1A1HPGDTP53SMN1; SMN2HSD17B10
SCHEMBL4347023 0.74 KMT2A (0.53) ALDH1A1HPGDSMN1; SMN2MAPTNPSR1
SCHEMBL27598146 0.74 ALDH1A1 (0.51) ALDH1A1MAPK1HPGDTP53TSHR
SCHEMBL4347093 0.73 RAB9A (0.47) ALDH1A1HPGDSMN1; SMN2L3MBTL1MAPT
SCHEMBL4345489 0.73 CA12 (0.47) ALDH1A1MAPTCA12CA1CA2
SCHEMBL11808657 0.72 TSHR (0.46) ALDH1A1MAPK1HPGDTSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed