SCHEMBL435758

SCHEMBL435758

Clc1ccc(-c2cc[c]cc2Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 3/20 0.42
CYP1A2 P05177 1/20 0.36
CYP2A6 P11509 2/20 0.35
LMNA P02545 1/20 0.35
PTGS2 P35354 3/20 0.34
TDO2 P48775 1/20 0.33
SRD5A2 P31213 1/20 0.33
PTGS1 P23219 1/20 0.32
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31
NFKB1 P19838 1/20 0.31
CASP3 P42574 1/20 0.31
RAB9A P51151 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
SENP8 Q96LD8 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2012244 0.83 PTGS2 (0.39) CYP2A6LMNAPTGS2TDO2PTGS1
SCHEMBL28822926 0.83 MAPK1 (0.33) CYP1A2CYP2A6LMNAALDH1A1TP53
SCHEMBL5899213 0.83 HPGD (0.35) CYP2A6PTGS2KDM4EALDH1A1HSD17B10
SCHEMBL21723073 0.83 AHR (0.42) AHRCYP1A2CYP2A6LMNAPTGS2
SCHEMBL2093448 0.83 CYP2A6 (0.54) CYP1A2CYP2A6LMNAKDM4EALDH1A1
SCHEMBL1135190 0.81
SCHEMBL27555403 0.81 CYP2A6 (0.52) CYP1A2CYP2A6LMNAKDM4EALDH1A1
SCHEMBL9067366 0.79 AHR (0.52) AHRKDM4ENPC1ALDH1A1TP53
SCHEMBL8506861 0.79 AHR (0.35) AHRCYP1A2CYP2A6LMNAPTGS2
SCHEMBL16720203 0.79 ALOX5 (0.41) AHRCYP1A2CYP2A6LMNAPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106047985-A High throughput screening method of alcohol dehydrogenase 江南大学 2016-10-26 CN claimed
US-8026085-B2 Methods and systems for selective fluorination of organic molecules CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2011-09-27 US claimed
CN-116583180-A Lactam composition and use 联合利华知识产权控股有限公司 2023-08-11 CN disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2004030671-A2 USE OF 4-AMINO-QUINAZOLINES AS ANTI CANCER AGENTS MERCK PATENT GMBH (DE) 2004-04-15 WO disclosed
WO-2004030672-A1 USE OF 4 AMINO-QUINAZOLINES AS ANTI CANCER AGENTS MERCK PATENT GMBH (DE) 2004-04-15 WO disclosed
EP-0363223-A2 3-Aryloxymethyl-cephalosporin derivatives, their preparation and their medical use Sankyo Company Limited (JP) 1990-04-11 EP disclosed