SCHEMBL4359741

SCHEMBL4359741

C=C1CCCC(C)(C)C1C(C)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.41
PTPN1 P18031 3/20 0.39
PTPN2 P17706 2/20 0.39
NR3C1 P04150 3/20 0.33
PGR P06401 3/20 0.33
AR P10275 3/20 0.33
NR3C2 P08235 1/20 0.33
PNLIP P16233 2/20 0.32
SOAT1 P35610 1/20 0.32
TDP1 Q9NUW8 2/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 2/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
STAT3 P40763 1/20 0.31
NLRP3 Q96P20 1/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2185238 0.85 TRPA1 (0.41) TRPA1PTPN1PTPN2NR3C1PGR
SCHEMBL11447720 0.81 PTPN1 (0.38) TRPA1PTPN1PTPN2NR3C1PGR
SCHEMBL11455730 0.81 PTPN1 (0.38) TRPA1PTPN1PTPN2PNLIPCYP3A4
SCHEMBL11316490 0.81 TRPA1 (0.36) TRPA1PTPN1PTPN2NR3C1PGR
SCHEMBL11447719 0.81 PTPN1 (0.38) TRPA1PTPN1PTPN2NR3C1PGR
SCHEMBL11447721 0.81 PTPN1 (0.38) TRPA1PTPN1PTPN2NR3C1PGR
SCHEMBL23530425 0.80 TRPA1 (0.39) TRPA1PTPN1PTPN2NR3C1PGR
SCHEMBL755859 0.80 TRPA1 (0.39) TRPA1PTPN1PTPN2NR3C1PGR
SCHEMBL17129801 0.80 TRPA1 (0.38) TRPA1PTPN1PTPN2NR3C1PGR
SCHEMBL29414123 0.80 TRPA1 (0.39) TRPA1PTPN1PTPN2NR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4268806-B2 2009-05-27 JP claimed
EP-1395542-B1 CATALYTIC SYSTEM FOR ALDOL REACTIONS FIRMENICH & CIE (CH) 2006-08-16 EP claimed
US-6838575-B2 Catalytic system for aldol reactions FIRMENICH SA (CH) 2005-01-04 US claimed
JP-2004529190-A 2004-09-24 JP claimed
US-20040082818-A1 Catalytic system for aldol reactions FIRMENICH SA (CH) 2004-04-29 US claimed
EP-1395542-A1 CATALYTIC SYSTEM FOR ALDOL REACTIONS FIRMENICH SA (CH) 2004-03-10 EP claimed
WO-2002094755-A1 CATALYTIC SYSTEM FOR ALDOL REACTIONS FIRMENICH SA (CH) 2002-11-28 WO claimed
EP-1697290-B1 PROCESS FOR THE ISOMERISATION OF A CYCLOHEXENYL ALKYL OR ALKENYL KETONE FIRMENICH & CIE (CH) 2012-09-12 EP disclosed
US-7250536-B2 Process for the isomerisation of a cyclohexenyl alkyl or alkenyl ketone FIRMENICH SA (CH) 2007-07-31 US disclosed
US-20060211889-A1 Process for the isomerisation of a cyclohexenyl alkyl or alkenyl ketone FIRMENICH SA (CH) 2006-09-21 US disclosed
EP-1697290-A1 PROCESS FOR THE ISOMERISATION OF A CYCLOHEXENYL ALKYL OR ALKENYL KETONE FIRMENICH SA (CH) 2006-09-06 EP disclosed
EP-1395542-B1 CATALYTIC SYSTEM FOR ALDOL REACTIONS FIRMENICH & CIE (CH) 2006-08-16 EP disclosed
US-7091151-B2 Catalytic system for aldol reactions FIRMENICH SA (CH) 2006-08-15 US disclosed
WO-2005061426-A1 PROCESS FOR THE ISOMERISATION OF A CYCLOHEXENYL ALKYL OR ALKENYL KETONE FIRMENICH SA (CH) 2005-07-07 WO disclosed
US-20050080297-A1 Group IV metal alkoxy halide complex and an alkyl or aryl carboxylic anhydride, BF3 or an anhydrous sulfate, chloride or bromide of Li+, Na+, K+, Cs+, Mg2+, Ni2+, Ca2+, Zn2+, Fe3+ or Al3+; for the one step aldol condensation of a ketone, e.g., a gem-dimethyl cyclohexylethanone with an aldehyde FIRMENICH SA (CH) 2005-04-14 US disclosed
US-6838575-B2 Catalytic system for aldol reactions FIRMENICH SA (CH) 2005-01-04 US disclosed
US-20040082818-A1 Catalytic system for aldol reactions FIRMENICH SA (CH) 2004-04-29 US disclosed
EP-1395542-A1 CATALYTIC SYSTEM FOR ALDOL REACTIONS FIRMENICH SA (CH) 2004-03-10 EP disclosed
WO-2002094755-A1 CATALYTIC SYSTEM FOR ALDOL REACTIONS FIRMENICH SA (CH) 2002-11-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050080297-A1 Group IV metal alkoxy halide complex and an alkyl or aryl carboxylic anhydride, BF3 or an anhydrous sulfate, chloride or bromide of Li+, Na+, K+, Cs+, Mg2+, Ni2+, Ca2+, Zn2+, Fe3+ or Al3+; for the one step aldol condensation of a ketone, e.g., a gem-dimethyl cyclohexylethanone with an aldehyde AKR1C3, CBR3, AKR1C2 TRPA1 899/4885PTPN1 4770/4885PTPN2 4722/4885
US-20060211889-A1 Process for the isomerisation of a cyclohexenyl alkyl or alkenyl ketone AKR1C3, AKR7A2, AKR1C2 TRPA1 2171/4885PTPN1 4664/4885PTPN2 4398/4885
US-20040082818-A1 Catalytic system for aldol reactions AKR1B10, AGL, AKR1C2 TRPA1 2394/4885PTPN1 4797/4885PTPN2 4766/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.