SCHEMBL4359785

SCHEMBL4359785

CCCc1nn(Cc2ccc(C(C)(C)C)cc2)c(=O)c(C(=O)NCC(=O)O)c1O

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGLN3 Q9H6Z9 10/20 0.68
KMT2A Q03164 1/20 0.50
EGLN1 Q9GZT9 11/20 0.47
EGLN2 Q96KS0 6/20 0.47
CYSLTR2 Q9NS75 1/20 0.43
PTGDR2 Q9Y5Y4 3/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
ATM Q13315 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4359892 0.89 EGLN3 (0.59) EGLN3EGLN1EGLN2CYSLTR2PTGDR2
SCHEMBL4362443 0.88 EGLN3 (0.52) EGLN3EGLN1EGLN2CYSLTR2PTGDR2
SCHEMBL3846940 0.86 EGLN3 (0.72) EGLN3KMT2AEGLN1EGLN2CYSLTR2
SCHEMBL4371854 0.85 EGLN3 (0.54) EGLN3EGLN1EGLN2CYSLTR2LMNA
SCHEMBL3857686 0.84 EGLN3 (0.93) EGLN3KMT2AEGLN1EGLN2CYSLTR2
SCHEMBL3850392 0.83 EGLN3 (0.69) EGLN3KMT2AEGLN1EGLN2CYSLTR2
SCHEMBL3847025 0.82 EGLN3 (0.86) EGLN3KMT2AEGLN1EGLN2CYSLTR2
SCHEMBL4359069 0.82 EGLN3 (0.51) EGLN3EGLN1EGLN2
SCHEMBL4363082 0.82 EGLN3 (0.51) EGLN3KMT2AEGLN1EGLN2LMNA
SCHEMBL3851851 0.81 EGLN3 (1.00) EGLN3KMT2AEGLN1EGLN2CYSLTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2124565-A2 N-SUBSTITUTED GLYCINE DERIVATIVES: HYDROXYLASE INHIBITORS Smithkline Beecham Corporation (US) 2009-12-02 EP claimed
WO-2008089052-A2 N-SUBSTITUTED GLYCINE DERIVATIVES: HYDROXYLASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-24 WO claimed