SCHEMBL4365804

SCHEMBL4365804

O=C(NSc1ccccc1OCc1cccc(C(F)(F)F)c1)NC(=O)c1cc2ccccc2o1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
GAA P10253 1/20 0.45
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
MAOB P27338 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SLC1A5 Q15758 1/20 0.40
PPIA P62937 1/20 0.40
ANO1 Q5XXA6 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
SIRT3 Q9NTG7 1/20 0.39
SLC6A4 P31645 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4365808 0.80 NPC1 (0.52) ALDH1A1L3MBTL1GAANFKB1NFKB2
SCHEMBL4369705 0.76 NPC1 (0.47) ALDH1A1NFKB1NFKB2RELANPC1
SCHEMBL4361842 0.76 NPC1 (0.46) ALDH1A1L3MBTL1GAANFKB1NFKB2
SCHEMBL13956851 0.75 MEN1 (0.57) ALDH1A1GAANFKB1NFKB2RELA
SCHEMBL4365813 0.74 MAPT (0.57) ALDH1A1GAANFKB1NFKB2RELA
SCHEMBL4361546 0.73 HPGD (0.49) ALDH1A1L3MBTL1GAANFKB1NFKB2
SCHEMBL4366956 0.73 SMN1; SMN2 (0.48) ALDH1A1NFKB1NFKB2RELANPC1
SCHEMBL3634482 0.69 SMN1; SMN2 (0.51) ALDH1A1NFKB1NFKB2RELANPC1
SCHEMBL4518242 0.69 NPC1 (0.43) ALDH1A1L3MBTL1GAANFKB1NFKB2
SCHEMBL4358710 0.68 RAB9A (0.47) ALDH1A1L3MBTL1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7476686-B2 Substituted aryl thioureas and related compounds; inhibitors of viral replication ACHILLION PHARMACEUTICALS, INC. (US) 2009-01-13 US claimed
US-20060014836-A1 Substituted aryl thioureas and related compounds; inhibitors of viral replication CHEN DAWEI 2006-01-19 US claimed
US-20040138205-A1 Substituted aryl thioureas and related compounds; inhibitors of viral replication ACHILLION PHARMACEUTICALS, INC. 2004-07-15 US claimed
US-7094807-B2 Substituted aryl thioureas and related compounds; inhibitors of viral replication ACHILLION PHARMACEUTICALS, INC. (US) 2006-08-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040138205-A1 Substituted aryl thioureas and related compounds; inhibitors of viral replication NAT1, PIGS, TPMT ALDH1A1 310/4885L3MBTL1 253/4885GAA 370/4885
US-20060014836-A1 Substituted aryl thioureas and related compounds; inhibitors of viral replication NAT1, PIGS, SLC10A1 ALDH1A1 221/4885L3MBTL1 168/4885GAA 407/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.