SCHEMBL436709

SCHEMBL436709

O=C(O)c1cccc2c1OCc1occ(F)c1-2

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
ALB P02768 1/20 0.37
HNF4A P41235 1/20 0.36
ALDH1A1 P00352 3/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
MYC P01106 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
HSD17B10 Q99714 1/20 0.34
NOTUM Q6P988 4/20 0.34
DHODH Q02127 3/20 0.32
HSP90AA1 P07900 1/20 0.32
ACMSD Q8TDX5 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436000 0.74 PARP1 (0.44) PARP1HNF4AALDH1A1L3MBTL1MYC
SCHEMBL20510040 0.71 PARP1 (0.73) PARP1HNF4AALDH1A1L3MBTL1MYC
SCHEMBL11094419 0.69 PARP1 (0.49) PARP1ALBALDH1A1MAPTHSD17B10
SCHEMBL14937360 0.64 PARP1 (0.41) PARP1HNF4AALDH1A1L3MBTL1MYC
SCHEMBL6836766 0.63 PARP1 (0.51) PARP1HNF4AALDH1A1L3MBTL1MYC
SCHEMBL20509570 0.63 PARP1 (0.37) PARP1ALBNPC1NOTUM
SCHEMBL16401466 0.62 MYC (0.61) ALBHNF4AALDH1A1L3MBTL1MYC
SCHEMBL31491647 0.62 ALB (0.47) ALBALDH1A1NPC1RAB9AHSD17B10
SCHEMBL19923221 0.61 HSD17B10 (0.59) ALBHNF4AALDH1A1L3MBTL1MYC
SCHEMBL69716 0.60 ALDH1A1 (0.69) ALBHNF4AALDH1A1L3MBTL1MYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595988-A1 TRICYCLIC COMPOUNDS AND METHDS OF MAKING AND USING SAME Zafgen, Inc. (US) 2013-05-29 EP disclosed
WO-2012012642-A1 TRICYCLIC COMPOUNDS AND METHDS OF MAKING AND USING SAME ZAFGEN CORPORATION (US) 2012-01-26 WO disclosed