SCHEMBL4368137

SCHEMBL4368137

Ic1cccc2cnccc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.59
CYP3A4 P08684 4/20 0.59
LMNA P02545 3/20 0.59
CYP2D6 P10635 3/20 0.59
CYP1A2 P05177 2/20 0.59
CYP2C19 P33261 2/20 0.59
CYP2C9 P11712 1/20 0.59
MAPKAPK2 P49137 1/20 0.59
HTT P42858 1/20 0.53
IKBKE Q14164 1/20 0.46
TBK1 Q9UHD2 1/20 0.46
ROCK2 O75116 2/20 0.44
ROCK1 Q13464 2/20 0.44
PIM1 P11309 1/20 0.43
HASPIN Q8TF76 1/20 0.43
KCNA3 P22001 1/20 0.42
IMPDH2 P12268 2/20 0.41
ALDH1A1 P00352 3/20 0.41
MAPT P10636 3/20 0.41
KMT2A Q03164 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30020533 1.00 KDM4E (0.59) KDM4ECYP3A4LMNACYP2D6CYP1A2
SCHEMBL18459080 0.83 TNF (0.53) KDM4ECYP3A4LMNACYP2D6CYP1A2
SCHEMBL29903107 0.83 TNF (0.53) KDM4ECYP3A4LMNACYP2D6CYP1A2
SCHEMBL18574399 0.77 KDM4E (0.42) KDM4ECYP3A4LMNACYP2D6CYP1A2
SCHEMBL6240424 0.77 LMNA (0.63) KDM4ECYP3A4LMNACYP2D6CYP1A2
SCHEMBL7948611 0.76 KDM4E (0.61) KDM4ECYP3A4LMNACYP2D6CYP1A2
SCHEMBL276517 0.74 CYP3A4 (0.59) KDM4ECYP3A4LMNACYP2D6CYP1A2
SCHEMBL12271 0.74 KDM4E (0.59) KDM4ECYP3A4LMNACYP2D6CYP1A2
SCHEMBL276518 0.74 KDM4E (1.00) KDM4ECYP3A4LMNACYP2D6CYP1A2
SCHEMBL3805113 0.74 CYP1A2 (0.59) KDM4ECYP3A4LMNACYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 206 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118190922-A Method for high-throughput screening of SARM1 inhibitor and application thereof 北京爱思益普生物科技股份有限公司 2024-06-14 CN claimed
CN-116496151-A Method for preparing fluorenone derivative by using Catellani strategy 长沙医学院 2023-07-28 CN claimed
CN-112300072-A High-yield synthesis method of 5-iodoisoquinoline compounds 常州工学院 2021-02-02 CN claimed
US-20260138987-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CONTINEUM THERAPEUTICS INC (US) 2026-05-21 US disclosed
US-12565501-B2 Muscarinic acetylcholine M1 receptor antagonists CONTINEUM THERAPEUTICS, INC. (US) 2026-03-03 US disclosed
EP-4613745-A2 PROCESS FOR PREPARING A COT INHIBITOR COMPOUND Gilead Sciences, Inc. (US) 2025-09-10 EP disclosed
US-12365666-B2 Process for preparing a Cot inhibitor compound GILEAD SCIENCES, INC. (US) 2025-07-22 US disclosed
CN-120283770-A Bacteriostat and application thereof in fruit disease control 中国科学院华南植物园 2025-07-11 CN disclosed
WO-2025129168-A1 TRIAZOLONE INHIBITORS OF NICOTINAMIDE N-METHYLTRANSFERASE AND THEIR THERAPEUTIC USES THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2025-06-19 WO disclosed
US-20250171455-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CONTINEUM THERAPEUTICS INC (US) 2025-05-29 US disclosed
EP-4126862-B1 PROCESS FOR PREPARING A COT INHIBITOR COMPOUND GILEAD SCIENCES INC (US) 2025-05-21 EP disclosed
EP-0872903-B1 Method for making hydrogen storage alloy powder and electrode comprising the alloy powder SHINETSU CHEMICAL CO (JP) 2001-10-04 EP disclosed
US-6277519-B1 QUENCHING AN ALLOY MELT; COMMINUTION SHIN-ETSU CHEMICAL CO., LTD. (JP) 2001-08-21 US disclosed
US-6096144-A TREATING WITH ACIDIC OR ALKALINE SOLUTION OF CONJUGATED UNSATURATED COMPOUND WITH AT LEAST 5 BONDS SHIN-ETSU CHEMICAL CO., LTD. (JP) 2000-08-01 US disclosed
US-5858571-A TREATING A PULVERIZED HYDROGEN ABSORBING ALLOY WITH A SOLUTION COMPRISING A CONJUGATED UNSATURATED COMPOUND SHIN-ETSU CHEMICAL CO., LTD. (JP) 1999-01-12 US disclosed
EP-0872903-A1 Method for making hydrogen storage alloy powder and electrode comprising the alloy powder Shin-Etsu Chemical Co., Ltd. (JP) 1998-10-21 EP disclosed
EP-0172427-B1 PROCESS FOR PRODUCTION OF VINYL CHLORIDE POLYMER Shin-Etsu Chemical Co., Ltd. (JP) 1989-07-05 EP disclosed
US-4758639-A Process for production of vinyl polymer SHIN-ETSU CHEMICAL CO., LTD. (JP) 1988-07-19 US disclosed
US-4757124-A Suspension or emulsion polymerizing vinyl chloride monomer or mixture of vinyl chloride with vinyl monomer copolymerizable therewith in reactor with walls coated with antiscaling compound containing dye or pigments SHIN-ETSU CHEMICAL CO., LTD. (JP) 1988-07-12 US disclosed
EP-0172427-A2 Process for production of vinyl chloride polymer Shin-Etsu Chemical Co., Ltd. (JP) 1986-02-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12565501-B2 Muscarinic acetylcholine M1 receptor antagonists CHRM1, CHRM2, CHRM3 KDM4E 3624/4885CYP3A4 1234/4885LMNA 3446/4885
US-12365666-B2 Process for preparing a Cot inhibitor compound TPO, TFPI, TFPI2 KDM4E 847/4885CYP3A4 784/4885LMNA 3342/4885
US-20260138987-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CHRM1, CHRM5, CHRM3 KDM4E 3909/4885CYP3A4 1239/4885LMNA 2976/4885
US-20250171455-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CHRM1, CHRM2, CHRM3 KDM4E 3057/4885CYP3A4 1279/4885LMNA 2924/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.