SCHEMBL4369696

SCHEMBL4369696

COc1cc2ncnc(Oc3ccc4oc(Nc5ccc(Cl)c(OC[C@@H]6CCCN6C)c5)nc4c3)c2cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDR P35968 16/20 1.00
LCK P06239 1/20 0.66
CSF1R P07333 1/20 0.66
IGF1R P08069 1/20 0.66
MET P08581 1/20 0.66
KIT P10721 1/20 0.66
FGFR1 P11362 1/20 0.66
SRC P12931 1/20 0.66
FGFR2 P21802 1/20 0.66
FGFR4 P22455 1/20 0.66
FGFR3 P22607 1/20 0.66
TEK Q02763 1/20 0.66
EPHA2 P29317 7/20 0.52
EPHB4 P54760 7/20 0.52
ERBB2 P04626 3/20 0.49
EGFR P00533 4/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4367877 1.00 KDR (1.00) KDRLCKCSF1RIGF1RMET
SCHEMBL4367282 0.90 KDR (1.00) KDRLCKCSF1RIGF1RMET
SCHEMBL4367190 0.90 KDR (1.00) KDRLCKCSF1RIGF1RMET
SCHEMBL4368103 0.85 KDR (0.74) KDRLCKCSF1RIGF1RMET
SCHEMBL4365198 0.85 KDR (0.74) KDRLCKCSF1RIGF1RMET
SCHEMBL4362208 0.82 KDR (0.82) KDRLCKCSF1RIGF1RMET
SCHEMBL13861963 0.82 KDR (0.82) KDRLCKCSF1RIGF1RMET
SCHEMBL4364745 0.81 KDR (0.80) KDRLCKCSF1RIGF1RMET
SCHEMBL4362982 0.81 KDR (1.00) KDRLCKCSF1RIGF1RMET
SCHEMBL4364757 0.80 KDR (0.75) KDRLCKCSF1RIGF1RMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7531553-B2 Heterocyclic compounds and methods of use AMGEN INC. (US) 2009-05-12 US disclosed
US-7531553-B2 Heterocyclic compounds and methods of use AMGEN INC. (US) 2009-05-12 US disclosed
US-7531553-B2 Heterocyclic compounds and methods of use AMGEN INC. (US) 2009-05-12 US disclosed
US-20040209892-A1 Heterocyclic compounds and methods of use U.S. PATENT OPERATIONS 2004-10-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040209892-A1 Heterocyclic compounds and methods of use VHL, NQO1, HPGDS KDR 83/4885LCK 1957/4885CSF1R 2626/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.