SCHEMBL4369739

SCHEMBL4369739

NC(=O)C(N)c1ccc(-c2cccnc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 10/20 0.61
MKNK2 Q9HBH9 10/20 0.61
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
CYP2A6 P11509 2/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
PARP1 P09874 1/20 0.47
DHODH Q02127 1/20 0.47
PARP2 Q9UGN5 1/20 0.47
LRRK2 Q5S007 1/20 0.45
DPP4 P27487 1/20 0.44
DPP7 Q9UHL4 1/20 0.44
KMO O15229 1/20 0.44
CHEK2 O96017 1/20 0.44
KIF11 P52732 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30338756 0.83 MKNK1 (0.59) MKNK1MKNK2CA12CA1CA2
SCHEMBL1354541 0.81 F7 (0.50) MKNK1MKNK2ALDH1A1
SCHEMBL1354543 0.81 F7 (0.50) MKNK1MKNK2ALDH1A1
SCHEMBL7193261 0.81 PTGS2 (0.52) DHODHDPP4
SCHEMBL2925473 0.79 MKNK1 (0.55) MKNK1MKNK2CA12CA1CA2
SCHEMBL6026 0.79 MKNK1 (0.55) MKNK1MKNK2CA12CA1CA2
SCHEMBL7237272 0.77 MKNK1 (0.54) MKNK1MKNK2CA12CA1CA2
SCHEMBL29337469 0.76 CYP2A6 (0.56) MKNK1MKNK2CA12CA1CA2
SCHEMBL606654 0.76 MKNK1 (1.00) MKNK1MKNK2CA12CA1CA2
SCHEMBL30855339 0.76 MKNK1 (1.00) MKNK1MKNK2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009012375-A2 SQUARATE KINASE INHIBITORS WYETH (US) 2009-01-22 WO disclosed