SCHEMBL437007

SCHEMBL437007

Brc1ccc2c(c1)C1(c3cc(Br)ccc3-2)c2cc(Br)ccc2-c2ccc(Br)cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.47
S100A4 P26447 1/20 0.44
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
TDP2 O95551 1/20 0.41
AKR1A1 P14550 1/20 0.41
AKR1B1 P15121 1/20 0.41
PTPRC P08575 1/20 0.38
METAP1 P53582 1/20 0.38
CYP2A6 P11509 2/20 0.37
BCL2 P10415 2/20 0.37
MCL1 Q07820 1/20 0.37
TGM2 P21980 1/20 0.35
CES1 P23141 1/20 0.35
KDM1A O60341 1/20 0.35
AHR P35869 2/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29404184 1.00 PDK2 (0.47) PDK2S100A4CA1CA2CA4
SCHEMBL29397249 0.89 PDK2 (0.58) PDK2S100A4CA1CA2CA4
SCHEMBL29399278 0.89 PDK2 (0.58) PDK2S100A4CA1CA2CA4
SCHEMBL29511719 0.89 PDK2 (0.58) PDK2S100A4CA1CA2CA4
SCHEMBL783463 0.89 PDK2 (0.58) PDK2S100A4CA1CA2CA4
SCHEMBL783450 0.89 PDK2 (0.58) PDK2S100A4CA1CA2CA4
SCHEMBL996751 0.89 PDK2 (0.58) PDK2S100A4CA1CA2CA4
SCHEMBL29574412 0.89 PDK2 (0.58) PDK2S100A4CA1CA2CA4
SCHEMBL29530902 0.89 PDK2 (0.58) PDK2S100A4CA1CA2CA4
SCHEMBL29602609 0.89 PDK2 (0.58) PDK2S100A4CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 209 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4406944-B1 SPIRO-TYPE HOLE TRANSPORT MATERIALS WITH EXTENDED EDGE PI-CONJUGATION LENGTH TOYOTA MOTOR CO LTD (JP) 2025-10-29 EP claimed
EP-4406944-A1 SPIRO-TYPE HOLE TRANSPORT MATERIALS WITH EXTENDED EDGE PI-CONJUGATION LENGTH TOYOTA JIDOSHA KABUSHIKI KAISHA (JP) 2024-07-31 EP claimed
CN-115505103-A Conjugated microporous polymer, and organic amine catalytic synthesis method and application thereof 华中科技大学 2022-12-23 CN claimed
CN-115286520-A Preparation method of hole transport material Spiro-OMeTAD 黑龙江省科学院石油化学研究院 2022-11-04 CN claimed
CN-110204696-B Sulfur-containing porous organic polymer material LNUs and preparation method and application thereof 辽宁大学 2022-03-29 CN claimed
CN-110256645-B Spherical covalent organic framework material and preparation method and application thereof 南京邮电大学 2021-10-26 CN claimed
CN-107917904-B Rapid detection Fe3+Method (2) 山东大学 2021-06-22 CN claimed
CN-107987093-B Small molecule taking spirobifluorene as core and preparation method thereof 武汉工程大学 2020-11-27 CN claimed
CN-110872261-A Organic semiconductor material substituted by oxadiazole containing spirofluorene, preparation method and OLED device 上海和辉光电有限公司 2020-03-10 CN claimed
US-9997714-B2 Hole transport material MERCK PATENT GMBH (DE) 2018-06-12 US claimed
US-20160254449-A1 HOLE TRANSPORT MATERIAL MERCK PATENT GMBH (DE) 2016-09-01 US claimed
EP-3052470-A1 HOLE TRANSPORT MATERIAL Merck Patent GmbH (DE) 2016-08-10 EP claimed
WO-2015049031-A1 HOLE TRANSPORT MATERIAL MERCK PATENT GMBH (DE) 2015-04-09 WO claimed
EP-4406944-B1 SPIRO-TYPE HOLE TRANSPORT MATERIALS WITH EXTENDED EDGE PI-CONJUGATION LENGTH TOYOTA MOTOR CO LTD (JP) 2025-10-29 EP disclosed
EP-4631926-A1 METHOD FOR PRODUCING HOMO-COUPLING REACTION PRODUCT National University Corporation Hokkaido University (JP) 2025-10-15 EP disclosed
EP-3169722-B9 NANOPARTICLES CHROMITION LTD (GB) 2025-06-18 EP disclosed
US-5840217-A LIGHT-EMITTING, CHARGE-TRANSPORT, CHARGE-INJECTION MATERIALS HOECHST AKTIENGESELLSCHAFT (DE) 1998-11-24 US disclosed
WO-1998018996-A1 OPTICAL BRIGHTENING AGENT AVENTIS RESEARCH & TECHNOLOGIES GMBH & CO KG (DE) 1998-05-07 WO disclosed
EP-0676461-A2 Spiro compounds and their application as electroluminescence materials HOECHST AKTIENGESELLSCHAFT (DE) 1995-10-11 EP disclosed
US-5026894-A Compound for use in the synthesis of semiconducting polymers with perpendicularly arranged cores and method of synthesizing said compound UNIVERSITY OF SOUTH CAROLINA (US) 1991-06-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160254449-A1 HOLE TRANSPORT MATERIAL SUN2, SLC6A19, SLCO2A1 PDK2 2494/4885S100A4 693/4885CA1 4821/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.