SCHEMBL4370773

SCHEMBL4370773

O=C(NSc1cccc(Cc2cccnc2)c1)NC(=O)c1cc2ccccc2o1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.56
TP53 P04637 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
CYP3A4 P08684 1/20 0.48
BLM P54132 1/20 0.48
HPGD P15428 2/20 0.46
KDM4E B2RXH2 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
CHRNB2 P17787 4/20 0.45
CHRNA7 P36544 4/20 0.45
CHRNA4 P43681 4/20 0.45
KCNH2 Q12809 1/20 0.45
GFER P55789 1/20 0.44
NPC1 O15118 1/20 0.43
LMNA P02545 1/20 0.43
TSHR P16473 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
PTK2B Q14289 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4368090 0.92 ALDH1A1 (0.56) ALDH1A1TP53MEN1KMT2AHPGD
SCHEMBL3634482 0.89 SMN1; SMN2 (0.51) ALDH1A1TP53MEN1KMT2AHPGD
SCHEMBL4366368 0.84 ALDH1A1 (0.50) ALDH1A1TP53MEN1KMT2AHPGD
SCHEMBL4366956 0.80 SMN1; SMN2 (0.48) ALDH1A1TP53MEN1KMT2AHPGD
SCHEMBL4370668 0.79 SMN1; SMN2 (0.50) ALDH1A1TP53MEN1KMT2AHPGD
SCHEMBL4370777 0.78 ALDH1A1 (0.77) ALDH1A1TP53MEN1KMT2ACYP3A4
SCHEMBL4375566 0.77 SMN1; SMN2 (0.49) ALDH1A1TP53MEN1KMT2AHPGD
SCHEMBL4361546 0.77 HPGD (0.49) ALDH1A1TP53MEN1KMT2AHPGD
SCHEMBL4360383 0.76 SMN1; SMN2 (0.47) ALDH1A1TP53MEN1KMT2AHPGD
SCHEMBL4365533 0.74 NPC1 (0.47) ALDH1A1TP53MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7476686-B2 Substituted aryl thioureas and related compounds; inhibitors of viral replication ACHILLION PHARMACEUTICALS, INC. (US) 2009-01-13 US claimed
US-20060014836-A1 Substituted aryl thioureas and related compounds; inhibitors of viral replication CHEN DAWEI 2006-01-19 US claimed
US-20040138205-A1 Substituted aryl thioureas and related compounds; inhibitors of viral replication ACHILLION PHARMACEUTICALS, INC. 2004-07-15 US claimed
US-7476686-B2 Substituted aryl thioureas and related compounds; inhibitors of viral replication ACHILLION PHARMACEUTICALS, INC. (US) 2009-01-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040138205-A1 Substituted aryl thioureas and related compounds; inhibitors of viral replication NAT1, PIGS, TPMT ALDH1A1 310/4885TP53 1296/4885MEN1 4797/4885
US-20060014836-A1 Substituted aryl thioureas and related compounds; inhibitors of viral replication NAT1, PIGS, SLC10A1 ALDH1A1 221/4885TP53 1070/4885MEN1 4762/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.