SCHEMBL4371697

SCHEMBL4371697

COc1cc(C(CCN(C)C)C2CC=CS2)ccc1OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.43
KMT2A Q03164 5/20 0.43
APP P05067 3/20 0.43
KDM4E B2RXH2 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
BLM P54132 1/20 0.42
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
F2 P00734 2/20 0.39
F10 P00742 2/20 0.39
PRSS1 P07477 2/20 0.39
F7 P08709 2/20 0.39
PRSS2 P07478 1/20 0.39
F3 P13726 1/20 0.39
PRSS3 P35030 1/20 0.39
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4366814 0.91 APP (0.39) MEN1KMT2AAPPKDM4ECYP1A2
SCHEMBL4372447 0.83 MEN1 (0.48) MEN1KMT2AAPPKDM4EGAA
SCHEMBL4371698 0.82 MEN1 (0.44) MEN1KMT2AAPPKDM4ECYP1A2
SCHEMBL4369064 0.78 APP (0.50) MEN1KMT2AAPPKDM4EPOLB
SCHEMBL4379009 0.74 SMN1; SMN2 (0.38) MEN1KMT2AKDM4EGAASMN1; SMN2
SCHEMBL4366818 0.72 APP (0.40) MEN1KMT2AAPPKDM4ECYP1A2
SCHEMBL12738664 0.71 NPC1 (0.55) MEN1KMT2AAPPKDM4ECYP1A2
SCHEMBL4375400 0.70 ALDH1A1 (0.39) MEN1KMT2APOLBSMN1; SMN2HPGD
SCHEMBL2999761 0.69 TNF (0.51) MEN1KMT2AKDM4ECYP1A2CYP3A4
SCHEMBL19734616 0.68 NPC1 (0.57) MEN1KMT2AAPPKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2083011-B1 PYRROLINE DERIVATIVES AGAINST CELL RELEASING TUMOR NECROSIS FACTOR, PREPARATION METHODS AND USES THEREOF TIANJIN HEMAY BIO TECH CO LTD (CN) 2014-06-04 EP disclosed
EP-2083011-A1 PYRROLINE DERIVATIVES AGAINST CELL RELEASING TUMOR NECROSIS FACTOR, PREPARATION METHODS AND USES THEREOF Tian Jin Hemay Bio-Tech Co., Ltd. (CN) 2009-07-29 EP disclosed