SCHEMBL4371981

SCHEMBL4371981

O=C(O)C[C@@H](c1ccc2c(n1)OC(=O)CN2)N1CCC(CCCc2ccc3c(n2)NCCC3)C1=O

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.64
ITGB3 P05106 18/20 0.64
ITGB5 P18084 1/20 0.47
ITGB6 P18564 3/20 0.46
ITGB8 P26012 3/20 0.46
ITGB1 P05556 1/20 0.46
ITGA2B P08514 1/20 0.46
ITGA5 P08648 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3884027 0.87 ITGB3 (0.76) ITGAVITGB3ITGB5ITGB1
SCHEMBL4370191 0.84 ITGB3 (0.76) ITGAVITGB3ITGB5ITGA2B
SCHEMBL4370498 0.84 ITGB3 (0.76) ITGAVITGB3ITGB5ITGA2B
SCHEMBL3885042 0.84 ITGB3 (0.66) ITGAVITGB3ITGB5ITGB1
SCHEMBL7936710 0.84 ITGAV (0.73) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL4381234 0.84 ITGAV (0.73) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL4371975 0.80 ITGB3 (0.41) ITGAVITGB3
SCHEMBL7945748 0.80 ITGAV (0.77) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL7945753 0.80 ITGAV (0.77) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL3889356 0.80 ITGAV (0.72) ITGAVITGB3ITGB5ITGB6ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047425-A4 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2009-04-22 EP disclosed
EP-1047425-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-11-02 EP disclosed
WO-1999030709-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed