Domperidone

Domperidone

SCHEMBL43729

O=c1[nH]c2ccccc2n1CCCN1CCC(n2c(=O)[nH]c3cc(Cl)ccc32)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2

The experimentally established mechanism targets of Domperidone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 known ✓ P14416 5/20 1.00
OPRM1 P35372 6/20 1.00
DRD3 P35462 5/20 1.00
SLC6A4 P31645 4/20 1.00
HTR1A P08908 4/20 1.00
CYP2D6 P10635 3/20 1.00
HTR2A P28223 3/20 1.00
HRH1 P35367 3/20 1.00
HTR2B P41595 3/20 1.00
USP2 O75604 2/20 1.00
CYP1A2 P05177 2/20 1.00
ADRA2A P08913 2/20 1.00
OPRK1 P41145 2/20 1.00
ADRA1D P25100 2/20 1.00
ADRA1A P35348 2/20 1.00
MEN1 O00255 1/20 1.00
SLC22A2 O15244 1/20 1.00
NR1I2 O75469 1/20 1.00
GMNN O75496 1/20 1.00
LMNA P02545 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Domperidone SCHEMBL29373565 1.00 OPRM1 (1.00) OPRM1DRD2DRD3SLC6A4HTR1A
SCHEMBL11509148 1.00 OPRM1 (1.00) OPRM1DRD2DRD3SLC6A4HTR1A
Domperidone SCHEMBL27988838 0.99 OPRM1 (0.98) OPRM1DRD2DRD3SLC6A4HTR1A
Domperidone SCHEMBL29177488 0.99 OPRM1 (0.98) OPRM1DRD2DRD3SLC6A4HTR1A
Domperidone SCHEMBL5569643 0.99 OPRM1 (0.98) OPRM1DRD2DRD3SLC6A4HTR1A
Domperidone SCHEMBL11506647 0.98 OPRM1 (0.96) OPRM1DRD2DRD3SLC6A4HTR1A
Water SCHEMBL11508184 0.97 DRD2 (0.94) OPRM1DRD2DRD3SLC6A4HTR1A
Water SCHEMBL11508185 0.97 DRD2 (0.94) OPRM1DRD2DRD3SLC6A4HTR1A
SCHEMBL11507685 0.95 DRD2 (0.90) OPRM1DRD2DRD3SLC6A4HTR1A
Domperidone SCHEMBL11507534 0.94 DRD2 (0.89) OPRM1DRD2DRD3SLC6A4HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 20286 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122094963-A Cardioprotective lipids and methods of use 2026-05-26 CN claimed
CN-122031470-A Application of domperidone in preparing pharmaceutical preparation for treating inflammatory dermatosis 中国药科大学 2026-05-15 CN claimed
CN-122004156-A Method for cultivating GCRV-resistant grass carp strain based on artificial gynogenesis 湖南师范大学 2026-05-12 CN claimed
US-12617809-B2 Cardioprotective lipid and method of use SIGNPATH PHARMA, INC. (US) 2026-05-05 US claimed
WO-2026090593-A2 RNA BIOMARKERS FOR USE IN BARRETT'S ESOPHAGUS CITY OF HOPE (US) 2026-04-30 WO claimed
US-20260092141-A1 SERIES OF POLYMERS HAVING PROPERTIES OF ACID-SENSITIVE DEGRADATION AND TEMPERATURE SENSITIVITY AND DRUG LOADING COMPOSITION THEREOF NANJING FANTAI CHEMICAL PHARMACEUTICAL RESEARCH INSTITUTE (CN) 2026-04-02 US claimed
US-20260083717-A1 FORMULATIONS CONTAINING DEUTERATED DOMPERIDONE CINDOME PHARMA INC (US) 2026-03-26 US claimed
US-12582601-B2 Orodispersible powder composition BIOPHARMA SYNERGIES, S.L. (ES) 2026-03-24 US claimed
US-20260069593-A1 METHODS FOR TREATING CANCER AMGEN INC (US) 2026-03-12 US claimed
US-12529704-B2 Methods for objective assessment of stress, early detection of risk for stress disorders, matching individuals with treatments, monitoring response to treatment, and new methods of use for drugs INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2026-01-20 US claimed
EP-0487674-A1 INJECTABLE SLOW-RELEASE GALENICAL. APLICACIONES FARMACEUTICAS (MX) 1992-06-03 EP claimed
WO-1992000735-A1 ROPINIROLE AND DOMPERIDONE FOR USE IN THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF PARKINSON'S DISEASE SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-01-23 WO claimed
CN-1057960-A DELAY GALENIC PARENTERAL FORM FOR INJECTION APLICACIONES FARMACEUTICAS (MX) 1992-01-22 CN claimed
WO-1991019485-A1 INJECTABLE SLOW-RELEASE GALENICAL APLICACIONES FARMACEUTICAS, S.A. DE C.V. (MX) 1991-12-26 WO claimed
EP-0454773-A1 NOVEL PRODRUG DERIVATIVES OF BIOLOGICALLY ACTIVE AGENTS CONTAINING HYDROXYL GROUPS OR NH-ACIDIC GROUPS Bundgaard, Hans (DK) 1991-11-06 EP claimed
WO-1990008128-A1 NOVEL PRODRUG DERIVATIVES OF BIOLOGICALLY ACTIVE AGENTS CONTAINING HYDROXYL GROUPS OR NH-ACIDIC GROUPS BUNDGAARD HANS (DK) 1990-07-26 WO claimed
WO-1989004179-A1 PHARMACEUTICAL FORMULATIONS FOR TRANSDERMAL ADMINISTRATION ALSO LABORATORI S.A.S. (IT) 1989-05-18 WO claimed
US-4772616-A DOMPERIDONE THE TEXAS A & M UNIVERSITY SYSTEM (US) 1988-09-20 US claimed
EP-0140789-A2 Use of peripherally selective dopamine antagonists for the preparation of a medicament for the topical treatment of ocular hypertension MERCK & CO. INC. (US) 1985-05-08 EP claimed
US-4066772-A ANTIEMETICS JANSSEN PHARMACEUTICA N.V. (BE) 1978-01-03 US claimed