SCHEMBL4373589

SCHEMBL4373589

COc1cc2nccc(Oc3ccc4nc(NC(=O)c5ccc(C(C)(C)C)cc5)sc4c3)c2cc1OC

nearest known ligand 0.66

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.66
FGFR2 P21802 5/20 0.65
KDR P35968 4/20 0.59
SCD O00767 8/20 0.57
MEN1 O00255 2/20 0.57
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
KMT2A Q03164 2/20 0.57
MAP3K5 Q99683 1/20 0.56
AXL P30530 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4379209 0.93 MET (0.70) METKDRSCDMEN1NPC1
SCHEMBL4379965 0.92 MET (0.65) METFGFR2KDRSCDMEN1
SCHEMBL4378894 0.91 MET (0.68) METFGFR2KDRSCDMEN1
SCHEMBL4372566 0.90 MET (0.67) METFGFR2KDRSCDMEN1
SCHEMBL4367748 0.90 SCD (0.68) METFGFR2KDRSCDMEN1
SCHEMBL4368604 0.90 MET (0.77) METKDRSCDMEN1NPC1
SCHEMBL4370551 0.86 MET (0.64) METFGFR2KDRSCDMEN1
SCHEMBL4373376 0.86 MET (0.66) METFGFR2KDRSCDMEN1
SCHEMBL13587170 0.86 AXL (0.71) METKDRSCDMEN1NPC1
SCHEMBL4379986 0.86 SCD (0.71) METKDRSCDMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7626030-B2 Compounds and methods of use AMGEN INC. (US) 2009-12-01 US disclosed
US-7626030-B2 Compounds and methods of use AMGEN INC. (US) 2009-12-01 US disclosed
US-7626030-B2 Compounds and methods of use AMGEN INC. (US) 2009-12-01 US disclosed
US-20050245547-A1 6-((6,7-Bis(methoxy)-4-quinolinyl)oxy)-N-(3-methylphenyl)-1-benzofuran-3-carboxamide;antiproliferative; -metastasis; -carcinogenic; -tumor; -inflammatory; -arthritic agents;hypotensive agents; myocardium necrosis; rheumatic diseases; tyrosine kinase inhibitors; antiallergens; asthma AMGEN INC. 2005-11-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050245547-A1 6-((6,7-Bis(methoxy)-4-quinolinyl)oxy)-N-(3-methylphenyl)-1-benzofuran-3-carboxamide;antiproliferative; -metastasis; -carcinogenic; -tumor; -inflammatory; -arthritic agents;hypotensive agents; myocardium necrosis; rheumatic diseases; tyrosine kinase inhibitors; antiallergens; asthma HGF, MET, HGFAC MET 2/4885FGFR2 77/4885KDR 90/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.