SCHEMBL4373709

SCHEMBL4373709

Cc1cc(-c2cccnc2)ccc1Nc1ncccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 4/20 0.49
TNIK Q9UKE5 2/20 0.49
ABL1 P00519 4/20 0.49
BCR P11274 3/20 0.49
MKNK1 Q9BUB5 1/20 0.49
MKNK2 Q9HBH9 1/20 0.49
PRKCA P17252 1/20 0.48
CYP2A6 P11509 2/20 0.47
RIPK2 O43353 1/20 0.46
RET P07949 1/20 0.46
KDR P35968 1/20 0.46
MAPK14 Q16539 1/20 0.46
SLC2A1 P11166 1/20 0.46
NPC1 O15118 1/20 0.45
PDGFRB P09619 1/20 0.45
PDGFRA P16234 1/20 0.45
FLT3 P36888 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13615433 0.81 MKNK1 (0.54) TNIKABL1MKNK1MKNK2CYP2A6
SCHEMBL22628286 0.76 ABL1 (0.70) KITABL1BCRPRKCAPDGFRB
SCHEMBL14506746 0.76 MKNK1 (0.61) ABL1MKNK1MKNK2CYP2A6RET
SCHEMBL12217607 0.74 MKNK1 (0.60) ABL1MKNK1MKNK2CYP2A6RET
SCHEMBL3860532 0.74 ABL1 (0.83) KITABL1BCRPRKCARET
SCHEMBL17666287 0.74 RAPGEF4 (0.55) KDRNPC1ALDH1A1CYP1A2
SCHEMBL13036623 0.73 CYP2A6 (0.62) MKNK1MKNK2CYP2A6SLC2A1ALDH1A1
SCHEMBL19575436 0.72 ABL1 (0.62) KITABL1BCRPRKCAPDGFRB
SCHEMBL22793758 0.72 ABL1 (0.70) KITABL1BCRMKNK1MKNK2
SCHEMBL30921131 0.72 ABL1 (0.58) KITABL1BCRMKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009109991-A2 NOVEL HYDRAZIDE CONTAINING TYROSINE KINASE INHIBITORS SUN PHARMA ADVANCED RESEARCH COMPANY LTD., (IN) 2009-09-11 WO disclosed