SCHEMBL4376091

SCHEMBL4376091

Nc1nc(NCCc2cccs2)ncc1CCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 9/20 0.49
ADORA2A P29274 8/20 0.49
ADORA2B P29275 8/20 0.49
ADORA3 P0DMS8 6/20 0.49
APP P05067 1/20 0.44
FLT3 P36888 1/20 0.43
HTR2C P28335 1/20 0.41
HTR7 P34969 1/20 0.41
HTR6 P50406 1/20 0.41
IGF1R P08069 1/20 0.40
TMIGD3 P0DMS9 2/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
HIF1A Q16665 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4374779 0.77 ADORA2A (0.50) ADORA1ADORA2AADORA2BADORA3FLT3
SCHEMBL4376249 0.77 APP (0.46) APPKMT2AMEN1HDAC3HDAC1
SCHEMBL1091872 0.75 APP (0.50) ADORA1ADORA2AADORA2BADORA3APP
SCHEMBL7016043 0.73 APP (0.58) APPHDAC3HDAC1HDAC2HDAC6
SCHEMBL4376506 0.73 MEN1 (0.44) ADORA1ADORA2AADORA2BADORA3KMT2A
SCHEMBL4374733 0.72 ADORA2A (0.51) ADORA1ADORA2AADORA2BADORA3APP
SCHEMBL4376041 0.71 APP (0.49) ADORA1ADORA2AADORA2BADORA3APP
SCHEMBL4376781 0.71 APP (0.49) ADORA1ADORA2AADORA2BADORA3APP
SCHEMBL14869658 0.71 HTR6 (0.62) ADORA1ADORA2AADORA2BADORA3FLT3
SCHEMBL4377864 0.70 APP (0.48) ADORA1ADORA2AADORA2BAPPTMIGD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1280781-B1 5-HT 7 RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2009-11-18 EP disclosed