SCHEMBL4376249

SCHEMBL4376249

Nc1nc(NCc2ccncc2)ncc1CCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.46
KCNH3 Q9ULD8 2/20 0.46
ABCB1 P08183 2/20 0.44
BACE1 P56817 1/20 0.43
MAPT P10636 1/20 0.42
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016043 0.85 APP (0.58) APPHDAC3HDAC1HDAC2HDAC6
SCHEMBL1090705 0.81 HDAC1 (0.39) KCNH3HDAC3HDAC1HDAC2HDAC6
SCHEMBL4377159 0.81 APP (0.47) APPKCNH3ABCB1MEN1ALDH1A1
SCHEMBL4376091 0.77 ADORA1 (0.49) APPMEN1KMT2AHDAC3HDAC1
SCHEMBL7011552 0.76 LTA4H (0.46) MEN1ALDH1A1KMT2AHDAC3HDAC1
SCHEMBL3447051 0.75 CSF1R (0.47)
SCHEMBL1317138 0.74 DHFR (0.54)
SCHEMBL7013050 0.73 HTR7 (0.53) HDAC3HDAC1HDAC2HDAC6
SCHEMBL1090916 0.73 CHRNA7 (0.52) MEN1ALDH1A1KMT2AHDAC3HDAC1
SCHEMBL4376349 0.72 APP (0.52) APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1280781-B1 5-HT 7 RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2009-11-18 EP claimed