Formamide

Formamide

SCHEMBL4376802

CC1Cc2ccccc2N1C.NC=O

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.50
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
KMT2A Q03164 1/20 0.44
LMNA P02545 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
ROCK1 Q13464 1/20 0.41
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
HTR2A P28223 3/20 0.41
HTR2C P28335 3/20 0.41
HTR2B P41595 3/20 0.41
NPC1 O15118 2/20 0.40
ALDH1A1 P00352 2/20 0.40
PKM P14618 1/20 0.40
RAB9A P51151 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7733992 0.89 NOTUM (0.55) NOTUMMEN1MAPTKMT2ALMNA
SCHEMBL811795 0.89 NOTUM (0.55) NOTUMMEN1MAPTKMT2ALMNA
SCHEMBL6890897 0.89 NOTUM (0.55) NOTUMMEN1MAPTKMT2ALMNA
SCHEMBL31672940 0.89 NOTUM (0.55) NOTUMMEN1MAPTKMT2ALMNA
Ammonia Solution, Strong SCHEMBL29093479 0.87 NOTUM (0.53) NOTUMMEN1MAPTKMT2ALMNA
Hydrochloric Acid SCHEMBL28861795 0.87 NOTUM (0.53) NOTUMMEN1MAPTKMT2ALMNA
SCHEMBL27711736 0.86 NOTUM (0.50) NOTUMMEN1MAPTKMT2ALMNA
SCHEMBL8516304 0.75 NOTUM (0.53) NOTUMMEN1MAPTKMT2ALMNA
SCHEMBL23346693 0.72 AADAT (0.44) NOTUMHTR2AHTR2CHTR2B
SCHEMBL13070447 0.72 NOTUM (0.53) NOTUMMEN1MAPTKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115433116-B Acylated indoline derivative, composition and application thereof 徐州医科大学 2023-07-14 CN claimed
CN-115521302-A Tetrahydro (iso) quinoline or indoline derivative, composition and application thereof 徐州医科大学 2022-12-27 CN claimed
CN-115433116-A Acylated indoline derivative, composition and application thereof 徐州医科大学 2022-12-06 CN claimed
CN-115433116-B Acylated indoline derivative, composition and application thereof 徐州医科大学 2023-07-14 CN disclosed
CN-116249690-A Indoline compounds and derivatives as EGFR inhibitors 百济神州有限公司 2023-06-09 CN disclosed
CN-115894325-A Derivative containing aryl piperazine structure, composition and application thereof 徐州医科大学 2023-04-04 CN disclosed
CN-115521302-A Tetrahydro (iso) quinoline or indoline derivative, composition and application thereof 徐州医科大学 2022-12-27 CN disclosed
CN-115433116-A Acylated indoline derivative, composition and application thereof 徐州医科大学 2022-12-06 CN disclosed
CN-114748622-A P38 kinase inhibitors reduce DUX4 and downstream gene expression for the treatment of FSHD 弗尔康医疗公司 2022-07-15 CN disclosed
CN-114732910-A P38 kinase inhibitor reduces DUX4 and downstream gene expression for treatment of FSHD 弗尔康医疗公司 2022-07-12 CN disclosed
CN-111601593-B P38 kinase inhibitor reduces DUX4 and downstream gene expression for treatment of FSHD 弗尔康医疗公司 2022-04-15 CN disclosed
CN-111601593-A P38 kinase inhibitor reduces DUX4 and downstream gene expression for treatment of FSHD 弗尔康医疗公司 2020-08-28 CN disclosed
EP-2643311-A1 BICYCLIC GPR119 MODULATORS Lupin Limited (IN) 2013-10-02 EP disclosed
WO-2012069917-A1 BICYCLIC GPR119 MODULATORS LUPIN LIMITED (IN) 2012-05-31 WO disclosed
US-7629363-B2 antiinflammatory agent for treating asthma and chronic pulmonary inflammatory disease PFIZER INC (US) 2009-12-08 US disclosed
EP-1490064-B1 SUBSTITUTED PYRIDINONES AS MODULATORS OF P38 MAP KINASE PHARMACIA CORP (US) 2009-11-18 EP disclosed
EP-1490064-A1 SUBSTITUTED PYRIDINONES AS MODULATORS OF P38 MAP KINASE Pharmacia Corporation (US) 2004-12-29 EP disclosed
US-20040058964-A1 Substituted pyridinones PHARMACIA LLC 2004-03-25 US disclosed
WO-2003068230-A1 SUBSTITUTED PYRIDINONES AS MODULATORS OF P38 MAP KINASE PHARMACIA CORPORATION (US) 2003-08-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040058964-A1 Substituted pyridinones MAPK1, MAPK6, MAPK7 NOTUM 3993/4885MEN1 4261/4885MAPT 2803/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.