SCHEMBL4378312

SCHEMBL4378312

CCOc1ccc2c(c1)c(C(=O)C(=O)NC1CC1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl.COc1ccc2c(c1)c(C(=O)C(=O)NC1CC1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 4/20 0.42
GSK3B P49841 1/20 0.38
EDNRB P24530 3/20 0.38
EPHX2 P34913 2/20 0.38
PTGS2 P35354 2/20 0.37
LMNA P02545 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
F2RL3 Q96RI0 1/20 0.36
MEN1 O00255 1/20 0.36
RGS12 O14924 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36
NFKB1 P19838 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3008414 0.97 EPHX2 (0.40) PLA2G2AEPHX2LMNASMN1; SMN2F2RL3
SCHEMBL3000840 0.95 PLA2G2A (0.46) PLA2G2AGSK3BEPHX2PTGS2LMNA
SCHEMBL3003522 0.94 EPHX2 (0.39) PLA2G2AEPHX2LMNASMN1; SMN2F2RL3
SCHEMBL2992530 0.94 EPHX2 (0.39) PLA2G2AEPHX2LMNASMN1; SMN2F2RL3
SCHEMBL2998239 0.93 MAPT (0.39) PLA2G2AEPHX2LMNASMN1; SMN2MEN1
SCHEMBL2994490 0.92 PLA2G2A (0.44) PLA2G2AGSK3BEPHX2PTGS2LMNA
SCHEMBL3005938 0.92 PLA2G2A (0.44) PLA2G2AGSK3BEPHX2PTGS2LMNA
SCHEMBL3006204 0.92 PLA2G2A (0.44) PLA2G2AGSK3BEPHX2PTGS2LMNA
SCHEMBL3004632 0.87 PLA2G2A (0.41) PLA2G2ALMNAMEN1RGS12ALDH1A1
SCHEMBL3001744 0.87 SIGMAR1 (0.40) EPHX2LMNAMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed