SCHEMBL4379060

SCHEMBL4379060

COc1cc(CON)ccn1

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 3/20 0.68
LOX P28300 2/20 0.68
IDO1 P14902 15/20 0.49
AGXT P21549 11/20 0.49
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2092744 0.85 LOXL2 (0.67) LOXL2LOX
SCHEMBL2092739 0.81 LOXL2 (0.62) LOXL2LOX
SCHEMBL449200 0.81 LOXL2 (1.00) LOXL2LOX
Hydrochloric Acid SCHEMBL463199 0.79 LOXL2 (0.96) LOXL2LOX
SCHEMBL4018107 0.79 LOXL2 (0.59) LOXL2LOX
SCHEMBL19251359 0.79 LOXL2 (0.59) LOXL2LOX
SCHEMBL805488 0.79 LOXL2 (0.69) LOXL2LOX
SCHEMBL6218599 0.78 LOXL2 (0.73) LOXL2LOXCYP3A4
SCHEMBL130180 0.77 LOXL2 (0.67) LOXL2LOX
SCHEMBL2224895 0.77 LOXL2 (0.67) LOXL2LOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090298878-A1 OXIME COMPOUNDS AND THE USE THEREOF PURDUE PHARMA L.P. 2009-12-03 US disclosed
US-20090298878-A1 OXIME COMPOUNDS AND THE USE THEREOF PURDUE PHARMA L.P. 2009-12-03 US disclosed
US-20090298878-A1 OXIME COMPOUNDS AND THE USE THEREOF PURDUE PHARMA L.P. 2009-12-03 US disclosed
EP-2040698-A2 OXIME COMPOUNDS AND THE USE THEREOF SHIONOGI & CO., LTD. (JP) 2009-04-01 EP disclosed
WO-2008008398-A2 OXIME COMPOUNDS AND THE USE THEREOF SHIONOGI & CO., LTD. (JP) 2008-01-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090298878-A1 OXIME COMPOUNDS AND THE USE THEREOF KCNN4, CACNA1A, KCNN3 LOXL2 593/4885LOX 570/4885IDO1 305/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.