SCHEMBL4379239

SCHEMBL4379239

COc1cc2nccc(Oc3ccc4nc(NCc5ccc(C(F)(F)F)cc5)sc4c3)c2cc1OC

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MET P08581 2/20 0.59
CACNA1B Q00975 3/20 0.54
KDR P35968 6/20 0.52
FGFR2 P21802 3/20 0.48
PDGFRB P09619 1/20 0.47
PDGFRA P16234 1/20 0.47
RAB9A P51151 2/20 0.46
CD274 Q9NZQ7 1/20 0.46
AURKA O14965 1/20 0.46
LCK P06239 1/20 0.46
TEK Q02763 1/20 0.46
AURKB Q96GD4 1/20 0.46
CSNK1D P48730 1/20 0.45
AXL P30530 1/20 0.45
NPC1 O15118 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4381473 0.91 MET (0.61) METCACNA1BKDRPDGFRBPDGFRA
SCHEMBL4379130 0.90 MET (0.61) METCACNA1BKDRFGFR2PDGFRB
SCHEMBL4381327 0.88 MET (0.73) METKDRFGFR2PDGFRBPDGFRA
SCHEMBL4371493 0.87 MET (0.60) METKDRFGFR2PDGFRBPDGFRA
SCHEMBL4379351 0.87 MET (0.60) METKDRFGFR2PDGFRBPDGFRA
SCHEMBL4370557 0.87 MET (0.60) METCACNA1BKDRFGFR2PDGFRB
SCHEMBL4371282 0.84 MET (0.61) METKDRFGFR2PDGFRBPDGFRA
SCHEMBL4366758 0.84 MET (0.65) METKDRPDGFRBPDGFRARAB9A
SCHEMBL4379965 0.84 MET (0.65) METKDRFGFR2RAB9AAURKA
SCHEMBL4371210 0.83 MET (0.63) METKDRFGFR2PDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7626030-B2 Compounds and methods of use AMGEN INC. (US) 2009-12-01 US disclosed
US-7626030-B2 Compounds and methods of use AMGEN INC. (US) 2009-12-01 US disclosed
US-7626030-B2 Compounds and methods of use AMGEN INC. (US) 2009-12-01 US disclosed
US-20050245547-A1 6-((6,7-Bis(methoxy)-4-quinolinyl)oxy)-N-(3-methylphenyl)-1-benzofuran-3-carboxamide;antiproliferative; -metastasis; -carcinogenic; -tumor; -inflammatory; -arthritic agents;hypotensive agents; myocardium necrosis; rheumatic diseases; tyrosine kinase inhibitors; antiallergens; asthma AMGEN INC. 2005-11-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050245547-A1 6-((6,7-Bis(methoxy)-4-quinolinyl)oxy)-N-(3-methylphenyl)-1-benzofuran-3-carboxamide;antiproliferative; -metastasis; -carcinogenic; -tumor; -inflammatory; -arthritic agents;hypotensive agents; myocardium necrosis; rheumatic diseases; tyrosine kinase inhibitors; antiallergens; asthma HGF, MET, HGFAC MET 2/4885CACNA1B 4597/4885KDR 90/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.