SCHEMBL4380282

SCHEMBL4380282

COc1ccc2c(c1)c(C(=O)C(=O)Nc1cccc(Cl)c1)c(C)n2Cc1ccc(Cl)cc1Cl.COc1cccc(NC(=O)C(=O)c2c(C)n(Cc3ccc(Cl)cc3Cl)c3ccc(OC)cc23)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.51
PLA2G2A P14555 7/20 0.49
MAPT P10636 5/20 0.48
THRB P10828 1/20 0.46
PTGER3 P43115 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
PKM P14618 2/20 0.44
HTT P42858 1/20 0.44
LMNA P02545 2/20 0.44
PTGS2 P35354 1/20 0.43
RGS12 O14924 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2170586 0.98 FAAH (0.53) FAAHPLA2G2AMAPTTHRBMEN1
SCHEMBL2159594 0.98 FAAH (0.53) FAAHPLA2G2AMAPTTHRBPTGER3
SCHEMBL2168611 0.92 PLA2G2A (0.56) FAAHPLA2G2AMAPTMEN1KMT2A
SCHEMBL3001541 0.91 PTGER3 (0.45) FAAHPLA2G2AMAPTPTGER3SMN1; SMN2
SCHEMBL3006040 0.91 PLA2G2A (0.44) FAAHPLA2G2AMAPTTHRBSMN1; SMN2
SCHEMBL2168630 0.89 FAAH (0.64) FAAHPLA2G2AMAPTMEN1KMT2A
SCHEMBL3001888 0.88 MAPT (0.46) FAAHMAPTPTGER3SMN1; SMN2NPC1
SCHEMBL2169000 0.88 FAAH (0.51) FAAHPLA2G2AMAPTMEN1KMT2A
SCHEMBL2159618 0.88 FAAH (0.60) FAAHPLA2G2AMAPTSMN1; SMN2MEN1
SCHEMBL2168110 0.88 FAAH (0.65) FAAHPLA2G2AMAPTSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed