SCHEMBL438098

SCHEMBL438098

c1ccc(CC2=C(Cc3ccccc3)CCCCC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CALM1 P0DP23 1/20 0.52
POLB P06746 1/20 0.44
TSHR P16473 1/20 0.43
LTA4H P09960 5/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
IDH1 O75874 1/20 0.40
PARP11 Q9NR21 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
DPP7 Q9UHL4 2/20 0.39
PLA2G10 O15496 1/20 0.39
PLA2G2A P14555 1/20 0.39
LMNA P02545 1/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19306461 1.00 CALM1 (0.52) CALM1POLBTSHRLTA4HL3MBTL1
SCHEMBL21807128 1.00 CALM1 (0.52) CALM1POLBTSHRLTA4HL3MBTL1
Hydrochloric Acid SCHEMBL11638839 0.88 LOXL2 (0.43) CALM1POLBLTA4HL3MBTL1PLA2G10
SCHEMBL9566501 0.87 CALM1 (0.61) CALM1TSHRLTA4HIDH1LMNA
SCHEMBL7752320 0.85 IDH1 (0.42) CALM1POLBIDH1DPP7PLA2G10
Hydrochloric Acid SCHEMBL11522917 0.83 IDH1 (0.41) CALM1POLBIDH1DPP7PLA2G10
SCHEMBL16322334 0.82 TP53 (0.46) CALM1TSHRLTA4HLMNA
Diphenylmethane SCHEMBL28085719 0.81 CALM1 (0.80) CALM1LTA4HIDH1HRH3PLA2G10
Diphenylmethane SCHEMBL28072604 0.81 CALM1 (0.80) CALM1LTA4HIDH1HRH3PLA2G10
SCHEMBL9806319 0.81 CALM1 (0.42) CALM1POLBTSHRLTA4HL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140171436-A1 TREATMENT OF ANTIFOLATE NEUROTOXICITY SYNTRIX BIOSYSTEMS, INC. (US) 2014-06-19 US disclosed
US-8101635-B2 Use of glutamate antagonists which is a NMDA receptor antagonist ( ifenprodil, memantine) to reduce or control retinal pigment epithelium and/or glial migration and the subsequent development of proliferative vitreoretinopathy ( vision defect ) ALLERGAN, INC. (US) 2012-01-24 US disclosed
US-20080193502-A1 MEMANTINE INTRAVITREAL IMPLANTS ALLERGAN, INC. (US) 2008-08-14 US disclosed
US-20080193503-A1 MEMANTINE INTRAVITREAL IMPLANTS ALLERGAN, INC. (US) 2008-08-14 US disclosed
US-20070148208-A1 ANTI-EXCITITOXIC SUSTAINED RELEASE INTRACULAR IMPLANTS AND RELATED METHODS ALLERGAN, INC. 2007-06-28 US disclosed
US-20070141117-A1 ANTI-EXCITITOXIC SUSTAINED RELEASE INTRAOCULAR IMPLANTS AND RELATED METHODS ALLERGAN, INC. 2007-06-21 US disclosed
US-7230032-B2 Calcium blockers to treat proliferative vitreoretinopathy ALLERGAN, INC. (US) 2007-06-12 US disclosed
CN-1950069-A Anti-excititoxic sustained release intracular implants and related methods ALLERGAN INC (US) 2007-04-18 CN disclosed
US-20050244478-A1 Anti-excititoxic sustained release intraocular implants and related methods ALLERGAN, INC. (US) 2005-11-03 US disclosed
US-20050244473-A1 Memantine intravitreal implants ALLERGAN, INC. (US) 2005-11-03 US disclosed
US-20050009884-A1 Calcium blockers to treat proliferative retinal diseases ALLERGAN, INC. 2005-01-13 US disclosed
US-20040266808-A1 Utilizing N-methyl-D-aspartate (NMDA) receptor antagonist at levels without side effects; uncompetitive open channel blocking SYNTRIX BIOSYSTEMS, INC. 2004-12-30 US disclosed
US-6573280-B2 Glutamate causes migration and proliferation of retinal pigment epithelium and/or glial cells, and glutamate antagonists can prevent, treat or reduce retinal pigment epithelium and/or glial migration and the subsequent ALLERGAN, INC. 2003-06-03 US disclosed
EP-0797442-B1 TREATMENT OF OPTIC NEURITIS MASSACHUSETTS EYE & EAR INFIRM (US) 2003-05-21 EP disclosed
US-6482854-B1 Glaucoma treatment MASSACHUSETTS EYE AND EAR INFIRMARY 2002-11-19 US disclosed
EP-0797442-A4 TREATMENT OF OPTIC NEURITIS MASSACHUSETTS EYE & EAR INFIRM (US) 1998-04-15 EP disclosed
EP-0797442-A1 TREATMENT OF OPTIC NEURITIS MASSACHUSETTS EYE & EAR INFIRMARY (US) 1997-10-01 EP disclosed
US-5597809-A METHYL ASPARTATE MEDIATED RETINAL CELL DAMAGE MASSACHUSETTS EYE & EAR INFIRMARY (US) 1997-01-28 US disclosed
WO-1996000073-A1 TREATMENT OF OPTIC NEURITIS MASSACHUSETTS EYE AND EAR INFIRMARY (US) 1996-01-04 WO disclosed
EP-0338532-A2 N-alkylamino derivates of aromatic, tricyclic compounds in the treatment of drug-resistant protozoal infections MERRELL DOW PHARMACEUTICALS INC. (US) 1989-10-25 EP disclosed