SCHEMBL4381898

SCHEMBL4381898

Cc1ccc2c(c1)c(C(=O)C(=O)NC1CCCCC1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1.O=C(NC1CCCCC1)C(=O)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccc(O)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 2/20 0.43
CNR2 P34972 3/20 0.42
HTT P42858 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TP53 P04637 4/20 0.41
S1PR3 Q99500 1/20 0.41
MAPT P10636 4/20 0.40
PKM P14618 3/20 0.40
GAA P10253 3/20 0.40
ALDH1A1 P00352 1/20 0.40
KDM4E B2RXH2 2/20 0.40
LMNA P02545 2/20 0.38
CNR1 P21554 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3006611 0.96 FAAH (0.46) FAAHCNR2HTTMEN1KMT2A
SCHEMBL3005497 0.95 FAAH (0.46) FAAHCNR2HTTMEN1KMT2A
SCHEMBL3005859 0.95 S1PR3 (0.44) FAAHCNR2HTTTP53S1PR3
SCHEMBL2996457 0.94 S1PR3 (0.44) CNR2HTTMEN1KMT2ATP53
SCHEMBL4391954 0.93 FAAH (0.45) FAAHCNR2HTTMEN1KMT2A
SCHEMBL3006284 0.93 FAAH (0.46) FAAHCNR2HTTMEN1KMT2A
SCHEMBL3010320 0.92 S1PR3 (0.42) FAAHHTTMEN1KMT2ATP53
SCHEMBL2999872 0.92 FAAH (0.47) FAAHCNR2HTTMEN1KMT2A
SCHEMBL3001499 0.91 S1PR3 (0.42) FAAHCNR2HTTMEN1KMT2A
SCHEMBL4386783 0.90 FAAH (0.46) FAAHCNR2HTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed