SCHEMBL4386783

SCHEMBL4386783

Cc1ccc2c(c1)c(C(=O)C(=O)NC1CC1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1.O=C(NC1CC1)C(=O)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccc(Cl)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.46
MEN1 O00255 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42
CNR2 P34972 4/20 0.41
TP53 P04637 3/20 0.37
PLA2G2A P14555 1/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
HIF1A Q16665 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PTGES2 Q9H7Z7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PPARG P37231 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2999872 0.98 FAAH (0.47) FAAHMEN1HTTKMT2ACNR2
SCHEMBL4391954 0.96 FAAH (0.45) FAAHMEN1HTTKMT2ACNR2
SCHEMBL3005497 0.94 FAAH (0.46) FAAHMEN1HTTKMT2ACNR2
SCHEMBL3006284 0.94 FAAH (0.46) FAAHMEN1HTTKMT2ACNR2
SCHEMBL3000962 0.94 CNR2 (0.41) FAAHMEN1KMT2ACNR2PLA2G2A
SCHEMBL3006611 0.94 FAAH (0.46) FAAHMEN1HTTKMT2ACNR2
SCHEMBL3006187 0.91 CNR2 (0.41) FAAHMEN1KMT2ACNR2TP53
SCHEMBL3005482 0.91 CNR2 (0.42) FAAHKMT2ACNR2TP53UBE2M
SCHEMBL4381898 0.90 FAAH (0.43) FAAHMEN1HTTKMT2ACNR2
SCHEMBL3008931 0.90 POLB (0.44) FAAHKMT2ACNR2TP53UBE2M

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed