SCHEMBL4382416

SCHEMBL4382416

CCC(CCCc1c[nH]cn1)OC(N)=O

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.33
PRKCD Q05655 1/20 0.33
MAP3K7 O43318 1/20 0.31
TAB1 Q15750 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4385034 0.91 PRKCA (0.33) PRKCAPRKCD
SCHEMBL4381434 0.89 HRH3 (0.34)
SCHEMBL4379173 0.88 PRKCA (0.34) PRKCAPRKCD
SCHEMBL4387568 0.86 HRH3 (0.35)
SCHEMBL4387281 0.86 HRH3 (0.35)
SCHEMBL8798625 0.85 CTSK (0.32) PRKCAPRKCD
SCHEMBL5157590 0.83 PRKCA (0.33) PRKCAPRKCD
SCHEMBL4386649 0.82
SCHEMBL4385037 0.79 HRH3 (0.36)
SCHEMBL8798303 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760811-B1 IMIDAZOLE DERIVATIVES AS HISTAMINE RECEPTOR H3 MODULATORS INST NAT SANTE RECH MED (FR) 2009-11-18 EP disclosed
US-6248765-B1 ANTIINFLAMMATORY AGENTS; HYPOTENSIVE AGENTS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICAL (FR) 2001-06-19 US disclosed
WO-1996029315-A2 IMIDAZOLE DERIVATIVES AS HISTAMINE RECEPTOR H3 (ANT)AGONISTS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 1996-09-26 WO disclosed