SCHEMBL4382829

SCHEMBL4382829

Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2c(c1)C(c1cccc(Cl)c1)SCc1nnnn1-2

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FNTA P49354 10/20 0.62
FNTB P49356 10/20 0.62
RORC P51449 4/20 0.41
PGGT1B P53609 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4374148 0.90 FNTA (0.63) FNTAFNTBPGGT1B
SCHEMBL4373656 0.85 FNTA (0.82) FNTAFNTBRORCPGGT1B
SCHEMBL4370606 0.85 FNTA (0.46) FNTAFNTBRORC
SCHEMBL1683552 0.83 FNTA (0.49) FNTAFNTBRORCPGGT1B
SCHEMBL6305116 0.82 FNTA (0.48) FNTAFNTBRORCPGGT1B
SCHEMBL4375776 0.80 FNTA (0.65) FNTAFNTBRORCPGGT1B
SCHEMBL4373631 0.79 FNTA (0.59) FNTAFNTBRORC
SCHEMBL4370392 0.79 FNTA (0.57) FNTAFNTBRORC
SCHEMBL4372579 0.79 FNTA (0.49) FNTAFNTBPGGT1B
SCHEMBL4384908 0.79 FNTA (0.55) FNTAFNTBRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339709-B1 FARNESYL TRANSFERASE INHIBITING BENZOHETEROCYCLIC DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2009-06-24 EP disclosed
US-7153958-B2 Farnesyl transferase inhibiting benzoheterocyclic derivatives JANSSEN PHARMACEUTICA N.V. (BE) 2006-12-26 US disclosed