SCHEMBL4384644

SCHEMBL4384644

COc1ccc2c(c1)CCN(CCCCl)C2

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.59
SLC6A2 P23975 3/20 0.58
SLC6A4 P31645 3/20 0.58
SLC6A3 Q01959 3/20 0.58
ABCB1 P08183 4/20 0.57
HRH3 Q9Y5N1 1/20 0.55
DRD1 P21728 1/20 0.55
DRD5 P21918 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3173969 0.86 ABCB1 (0.68) TDP1SLC6A2SLC6A4SLC6A3ABCB1
SCHEMBL22099626 0.86 SLC6A2 (0.55) TDP1SLC6A2SLC6A4SLC6A3ABCB1
SCHEMBL10675568 0.85 ABCB1 (0.67) TDP1SLC6A2SLC6A4SLC6A3ABCB1
SCHEMBL3246821 0.84 DRD1 (0.58) TDP1SLC6A2SLC6A4SLC6A3ABCB1
SCHEMBL3655159 0.83 HRH3 (0.61) SLC6A2SLC6A4SLC6A3ABCB1HRH3
SCHEMBL22099631 0.83 DRD1 (0.57) TDP1SLC6A2SLC6A4SLC6A3ABCB1
SCHEMBL915006 0.82 DRD1 (0.59) SLC6A2SLC6A4SLC6A3ABCB1DRD1
SCHEMBL29651184 0.82 DRD1 (0.59) SLC6A2SLC6A4SLC6A3ABCB1DRD1
SCHEMBL3245091 0.82 SLC6A4 (0.52) TDP1SLC6A2SLC6A4SLC6A3
SCHEMBL4390875 0.81 ABCB1 (0.74) SLC6A4ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144405-B1 TRIAZOLE COMPOUNDS WITH DOPAMINE-D3-RECEPTOR AFFINITY ABBOTT GMBH & CO KG (DE) 2009-11-25 EP disclosed
US-6602867-B1 Triazole compounds with dopamine-D3-receptor affinity ABBOTT LABORATORIES 2003-08-05 US disclosed