SCHEMBL4384764

SCHEMBL4384764

COc1cc2c(cc1OC)CN(CCCSc1nnc(-c3ccccc3)n1C)CC2

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 20/20 0.65
DRD2 P14416 18/20 0.65
HTR1A P08908 3/20 0.65
ADRA2C P18825 2/20 0.65
HRH2 P25021 2/20 0.65
ADRA1A P35348 2/20 0.65
HRH1 P35367 2/20 0.65
ADRA1B P35368 2/20 0.65
HTR2B P41595 2/20 0.65
ADRA2A P08913 1/20 0.65
ADRA2B P18089 1/20 0.65
DRD4 P21917 1/20 0.65
DRD5 P21918 1/20 0.65
HTR1B P28222 1/20 0.65
HTR2A P28223 1/20 0.65
HTR2C P28335 1/20 0.65
HTR7 P34969 1/20 0.65
CHRM2 P08172 1/20 0.60
CHRM4 P08173 1/20 0.60
CHRM3 P20309 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4387221 0.89 DRD3 (0.62) DRD3DRD2HTR1AADRA2CHRH2
SCHEMBL4378938 0.88 DRD3 (0.63) DRD3DRD2HTR1AADRA2CHRH2
SCHEMBL4381635 0.87 DRD3 (0.66) DRD3DRD2HTR1AADRA2CHRH2
SCHEMBL4389064 0.87 DRD3 (0.69) DRD3DRD2HTR1AADRA2CHRH2
SCHEMBL4390849 0.84 DRD3 (0.62) DRD3DRD2HTR1AADRA2CHRH2
Hydrochloric Acid SCHEMBL7201490 0.83 DRD3 (0.61) DRD3DRD2HTR1AADRA2CHRH2
SCHEMBL4382046 0.82 DRD3 (0.64) DRD3DRD2HTR1AHRH1KCNH2
SCHEMBL4380177 0.82 DRD3 (0.64) DRD3DRD2HTR1AHRH1KCNH2
SCHEMBL4389062 0.82 DRD3 (0.63) DRD3DRD2HTR1AADRA2CHRH2
Oxalic Acid SCHEMBL7204441 0.81 DRD3 (0.55) DRD3DRD2HTR1AADRA2CHRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144405-B1 TRIAZOLE COMPOUNDS WITH DOPAMINE-D3-RECEPTOR AFFINITY ABBOTT GMBH & CO KG (DE) 2009-11-25 EP disclosed
US-6602867-B1 Triazole compounds with dopamine-D3-receptor affinity ABBOTT LABORATORIES 2003-08-05 US disclosed