SCHEMBL4385684

SCHEMBL4385684

Cc1cc(COc2ccc(Nc3ncnc4cccc(OC[C@@H]5CCCN(C(=O)O)C5)c34)cc2Cl)no1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 17/20 0.56
EGFR P00533 11/20 0.56
KCNH2 Q12809 5/20 0.51
EPHA2 P29317 1/20 0.46
KDR P35968 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4540345 0.93 ERBB2 (0.62) ERBB2EGFRKCNH2
SCHEMBL5477568 0.92 ERBB2 (0.54) ERBB2EGFRKCNH2EPHA2KDR
SCHEMBL4384932 0.88 ERBB2 (0.72) ERBB2EGFRKCNH2
SCHEMBL4387752 0.88 ERBB2 (0.72) ERBB2EGFRKCNH2
SCHEMBL4390878 0.87 EGFR (0.63) ERBB2EGFRKCNH2
SCHEMBL4390260 0.87 EGFR (0.63) ERBB2EGFRKCNH2
SCHEMBL4385173 0.85 ERBB2 (0.53) ERBB2EGFRKCNH2EPHA2KDR
SCHEMBL4387569 0.85 ERBB2 (0.53) ERBB2EGFRKCNH2EPHA2KDR
SCHEMBL4385333 0.84 ERBB2 (0.79) ERBB2EGFRKCNH2
SCHEMBL5477579 0.84 ERBB2 (0.57) ERBB2EGFRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664029-B1 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2009-12-02 EP disclosed
EP-1664029-A1 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS AstraZeneca AB (SE) 2006-06-07 EP disclosed
WO-2005026152-A1 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2005-03-24 WO disclosed