SCHEMBL4387569

SCHEMBL4387569

O=C(O)N1CCC[C@H](COc2cccc3ncnc(Nc4ccc(O)c(Cl)c4)c23)C1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 11/20 0.53
EGFR P00533 9/20 0.53
SRC P12931 1/20 0.45
EPHA2 P29317 3/20 0.44
KDR P35968 3/20 0.44
EPHB4 P54760 2/20 0.44
KCNH2 Q12809 2/20 0.44
GRM5 P41594 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4385173 1.00 ERBB2 (0.53) ERBB2EGFRSRCEPHA2KDR
SCHEMBL5474052 0.90 ERBB2 (0.51) ERBB2EGFRSRCEPHA2KDR
SCHEMBL5479445 0.90 ERBB2 (0.51) ERBB2EGFRSRCEPHA2KDR
SCHEMBL4394667 0.87 EGFR (0.57) ERBB2EGFRSRCKCNH2
SCHEMBL4395377 0.87 EGFR (0.57) ERBB2EGFRSRCKCNH2
SCHEMBL4387752 0.87 ERBB2 (0.72) ERBB2EGFRKCNH2
SCHEMBL4384932 0.87 ERBB2 (0.72) ERBB2EGFRKCNH2
SCHEMBL4390878 0.85 EGFR (0.63) ERBB2EGFRKCNH2
SCHEMBL4390260 0.85 EGFR (0.63) ERBB2EGFRKCNH2
SCHEMBL4385684 0.85 ERBB2 (0.56) ERBB2EGFREPHA2KDRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664029-B1 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2009-12-02 EP disclosed