SCHEMBL4386792

SCHEMBL4386792

CC(=O)c1ccc2c(c1)CN(CCCSc1nnc(-c3ccc(C(F)(F)F)cc3)n1C)CC2

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 19/20 0.63
DRD2 P14416 17/20 0.63
KCNH2 Q12809 13/20 0.63
HRH1 P35367 1/20 0.59
CHRM1 P11229 2/20 0.55
CHRM3 P20309 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4387104 0.89 DRD3 (0.59) DRD3DRD2KCNH2HRH1
SCHEMBL4382046 0.84 DRD3 (0.64) DRD3DRD2KCNH2HRH1
SCHEMBL4702422 0.84 DRD3 (0.47) DRD3DRD2KCNH2
Hydrochloric Acid SCHEMBL7203533 0.84 DRD3 (0.63) DRD3DRD2KCNH2HRH1
SCHEMBL4703079 0.83 DRD3 (0.59) DRD3DRD2KCNH2
SCHEMBL4701629 0.81 DRD3 (0.59) DRD3DRD2KCNH2HRH1CHRM1
SCHEMBL4379086 0.81 DRD3 (0.52) DRD3DRD2KCNH2HRH1CHRM1
SCHEMBL4705240 0.81 DRD3 (0.58) DRD3DRD2KCNH2HRH1
SCHEMBL4380177 0.81 DRD3 (0.64) DRD3DRD2KCNH2HRH1
Hydrochloric Acid SCHEMBL7200726 0.81 DRD3 (0.51) DRD3DRD2KCNH2HRH1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144405-B1 TRIAZOLE COMPOUNDS WITH DOPAMINE-D3-RECEPTOR AFFINITY ABBOTT GMBH & CO KG (DE) 2009-11-25 EP claimed
EP-1144405-B1 TRIAZOLE COMPOUNDS WITH DOPAMINE-D3-RECEPTOR AFFINITY ABBOTT GMBH & CO KG (DE) 2009-11-25 EP disclosed
US-6602867-B1 Triazole compounds with dopamine-D3-receptor affinity ABBOTT LABORATORIES 2003-08-05 US disclosed