SCHEMBL4386845

SCHEMBL4386845

CC1=CC=CNC1[C@H]1CCC[C@@H](c2ncccc2C)N1CCCCNC(=O)c1ccc(O)nc1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.34
CYP19A1 P11511 1/20 0.34
KDM4E B2RXH2 1/20 0.33
DRD2 P14416 9/20 0.32
DRD3 P35462 9/20 0.32
DRD4 P21917 3/20 0.32
ADRA1A P35348 3/20 0.32
HTR1A P08908 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1B P35368 1/20 0.32
NAMPT P43490 1/20 0.32
SMYD2 Q9NRG4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2477001 0.87 ALDH1A1 (0.41) ALDH1A1CYP19A1KDM4EDRD2DRD3
SCHEMBL4390013 0.86 CXCR4 (0.38) KDM4E
SCHEMBL8305937 0.84 ALDH1A1 (0.44) ALDH1A1CYP19A1KDM4ESMYD2
SCHEMBL4239716 0.72 HDAC6 (0.37)
SCHEMBL2476696 0.72 CXCR4 (0.42) NAMPT
SCHEMBL2472935 0.71 CXCR4 (0.41) DRD2HTR1A
SCHEMBL2475481 0.70 CCR5 (0.45) DRD2DRD3
SCHEMBL8304298 0.70 ATM (0.40)
SCHEMBL11904802 0.70 CXCR4 (0.32)
SCHEMBL2472086 0.69 ATM (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7550484-B2 Chemokine receptor binding heterocyclic compounds with enhanced efficacy GENZYME CORPORATION (US) 2009-06-23 US claimed