SCHEMBL4387090

SCHEMBL4387090

O=S(=O)(c1ccc2c(c1)CN(CCCCl)CC2)N1CCOCC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.55
HTT P42858 2/20 0.48
BRD4 O60885 1/20 0.47
BRD2 P25440 1/20 0.47
BRD3 Q15059 1/20 0.47
ALDH1A1 P00352 5/20 0.46
GAA P10253 3/20 0.46
KDM4E B2RXH2 3/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
HPGD P15428 2/20 0.46
HSD17B10 Q99714 2/20 0.46
MAPT P10636 2/20 0.46
S1PR2 O95136 1/20 0.46
TNF P01375 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4770231 0.93 HTR2C (0.60) HTR2CHTTBRD4BRD2BRD3
SCHEMBL5098547 0.82 HTR2C (0.58) HTR2CBRD4ALDH1A1GAAKDM4E
SCHEMBL4392739 0.76 HTT (0.42) HTR2CHTTALDH1A1GAAKDM4E
Hydrochloric Acid SCHEMBL7199896 0.75 HTT (0.41) HTR2CHTTALDH1A1GAAKDM4E
SCHEMBL4380463 0.75 DRD3 (0.55) ALDH1A1KDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL4384867 0.73 MEN1 (0.40) HTR2CMEN1
SCHEMBL4394801 0.73 ALDH1A1 (0.60) HTR2CBRD4BRD2BRD3ALDH1A1
SCHEMBL4792242 0.73 HRH3 (0.48) PNMT
SCHEMBL4790927 0.72 HRH3 (0.47) HTR2CCYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL11467260 0.71 CA1 (0.51) PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144405-B1 TRIAZOLE COMPOUNDS WITH DOPAMINE-D3-RECEPTOR AFFINITY ABBOTT GMBH & CO KG (DE) 2009-11-25 EP disclosed
US-6602867-B1 Triazole compounds with dopamine-D3-receptor affinity ABBOTT LABORATORIES 2003-08-05 US disclosed