SCHEMBL4388997

SCHEMBL4388997

O=C(COc1ccc(OC(F)(F)F)cc1)NCc1nc(C(=O)NCc2ccccc2Cl)co1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 1/20 0.46
CACNA1H O95180 1/20 0.46
CACNA1I Q9P0X4 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
TRPV1 Q8NER1 1/20 0.46
SCN2A Q99250 2/20 0.45
SCN10A Q9Y5Y9 2/20 0.45
LMNA P02545 2/20 0.43
PLA2G1B P04054 1/20 0.42
POLB P06746 1/20 0.42
MAPK1 P28482 1/20 0.42
ATG4B Q9Y4P1 1/20 0.42
NPC1 O15118 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.40
MAPK8 P45983 2/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171264 0.88 NPC1 (0.55) CACNA1GCACNA1HCACNA1ISMN1; SMN2SCN2A
SCHEMBL5668902 0.87 CACNA1G (0.44) CACNA1GCACNA1HCACNA1ISMN1; SMN2SCN2A
SCHEMBL4392401 0.85 CACNA1G (0.51) CACNA1GCACNA1HCACNA1ISMN1; SMN2TRPV1
SCHEMBL2171492 0.85 TRPV1 (0.56) CACNA1GCACNA1HCACNA1ITRPV1SCN2A
SCHEMBL2173835 0.84 NPC1 (0.46) CACNA1GCACNA1HCACNA1ISMN1; SMN2SCN2A
SCHEMBL5668410 0.83 LTA4H (0.48) CACNA1GCACNA1HCACNA1ISMN1; SMN2TRPV1
SCHEMBL2172285 0.82 CACNA1G (0.45) CACNA1GCACNA1HCACNA1ISMN1; SMN2SCN10A
SCHEMBL4386435 0.81 CACNA1G (0.43) CACNA1GCACNA1HCACNA1IPOLBCYP1A2
SCHEMBL4394082 0.81 CACNA1G (0.43) CACNA1GCACNA1HCACNA1IPOLBCYP1A2
SCHEMBL2171605 0.80 TRPV1 (0.58) CACNA1GCACNA1HCACNA1ISMN1; SMN2TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090186905-A1 ANAPLASTIC LYMPHOMA KINASE MODULATORS AND METHODS OF USE EXELIXIS, INC. (US) 2009-07-23 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090186905-A1 ANAPLASTIC LYMPHOMA KINASE MODULATORS AND METHODS OF USE ALK, BCL3, MCL1 CACNA1G 4004/4885CACNA1H 4347/4885CACNA1I 4036/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.