SCHEMBL4389527

SCHEMBL4389527

CS(=O)(=O)NCc1ccc2c(n1)NCCC2

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 15/20 0.46
ITGB3 P05106 14/20 0.46
ITGB6 P18564 2/20 0.45
ITGB5 P18084 1/20 0.45
ITGB8 P26012 1/20 0.45
CXCR4 P61073 5/20 0.43
ITGA2B P08514 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31445490 0.84 ITGAV (0.57) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL4717885 0.79 CXCR4 (0.48) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL6921402 0.77 ITGAV (0.46) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL12895016 0.76 ITGAV (0.47) ITGAVITGB3ITGB6ITGB5CXCR4
SCHEMBL4389523 0.74 ITGAV (0.58) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL7797597 0.74 ITGAV (0.51) ITGAVITGB3ITGB6ITGB5CXCR4
SCHEMBL29416516 0.73 ITGAV (0.54) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL21328658 0.73 ITGAV (0.54) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL3138678 0.73 ITGAV (0.54) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL326631 0.73 ITGB3 (0.47) ITGAVITGB3ITGB6ITGB5ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049494-A2 TYROSINE KINASE INHIBITORS Merck & Co., Inc. (US) 2009-04-22 EP claimed
WO-2008008310-A2 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2008-01-17 WO claimed