SCHEMBL4389982

SCHEMBL4389982

Cc1c(N)ncnc1N1CCCCCC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.57
LMNA P02545 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
JAK3 P52333 2/20 0.50
NPC1 O15118 1/20 0.47
PKM P14618 1/20 0.47
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
MAP4K4 O95819 2/20 0.44
HTT P42858 3/20 0.44
ALOX15 P16050 1/20 0.44
AKT2 P31751 1/20 0.44
MAP3K5 Q99683 1/20 0.44
HSD17B10 Q99714 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
JAK2 O60674 1/20 0.42
IP6K1 Q92551 1/20 0.41
BTK Q06187 1/20 0.41
TP53 P04637 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17623135 0.82 KDM4E (0.70) LMNAJAK3KDM4EGAAMEN1
Hydrochloric Acid SCHEMBL31737655 0.81 HTR2C (0.53) ALDH1A1KDM4EGAAHTTMEN1
SCHEMBL20145916 0.78 RPS6KB1 (0.47) ALDH1A1LMNASMN1; SMN2JAK3NPC1
SCHEMBL9159049 0.76 HTT (0.61) ALDH1A1LMNASMN1; SMN2JAK3NPC1
SCHEMBL1871559 0.75 RPS6KB1 (0.50) ALDH1A1LMNASMN1; SMN2JAK3NPC1
SCHEMBL5889244 0.75 KDM4E (0.55) LMNASMN1; SMN2JAK3KDM4EGAA
SCHEMBL16071244 0.74 LRRK2 (0.54) ALDH1A1SMN1; SMN2JAK3KDM4EHTT
SCHEMBL10567632 0.74 LMNA (0.48) ALDH1A1LMNASMN1; SMN2JAK3NPC1
SCHEMBL11471053 0.73 HTT (0.58) ALDH1A1LMNASMN1; SMN2JAK3NPC1
Hydrochloric Acid SCHEMBL10567357 0.73 LMNA (0.47) ALDH1A1LMNASMN1; SMN2JAK3NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2117542-A1 COMBINATIONS OF BETA- 2 -ADRENOCEPTOR AGONISTIC BENZOTHIAZOLONE AstraZeneca AB (SE) 2009-11-18 EP disclosed
WO-2008096111-A1 COMBINATIONS OF BETA- 2 -ADRENOCEPTOR AGONISTIC BENZOTHIAZOLONE ASTRAZENECA AB (SE) 2008-08-14 WO disclosed