SCHEMBL4394419

SCHEMBL4394419

N#Cc1ccc(C(Cc2ccccc2)n2c(=O)[nH]c3cc(Cl)cc(Cl)c3c2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
MDM2 Q00987 4/20 0.39
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
GRIN1 Q05586 2/20 0.35
CYP19A1 P11511 2/20 0.34
MCHR1 Q99705 1/20 0.34
OPRM1 P35372 1/20 0.34
USP1 O94782 1/20 0.34
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
IDH1 O75874 1/20 0.33
FBP1 P09467 1/20 0.33
GPR17 Q13304 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4074600 0.85 ALK (0.41) SLC6A2SLC6A4
SCHEMBL4075249 0.77 CA12 (0.49) CA12CA9MDM2GRIN1OPRM1
SCHEMBL4211685 0.71 CA12 (0.52) CA12CA9GRIN1OPRM1USP1
SCHEMBL4223178 0.71 CA12 (0.52) CA12CA9GRIN1OPRM1USP1
SCHEMBL4214249 0.70 ALDH1A1 (0.57) CA12CA9GRIN1KDM4EMAPT
SCHEMBL4211671 0.67 CA12 (0.54) CA12CA9GRIN1KDM4EGAA
SCHEMBL4211573 0.66 CA12 (0.51) CA12CA9GRIN1KDM4EGAA
SCHEMBL13744898 0.66 MAPT (0.47) KDM4EMAPTL3MBTL1
SCHEMBL4217832 0.65 CA12 (0.60) CA12CA9GRIN1FBP1GPR17
SCHEMBL4220204 0.65 LMNA (0.57) CA12CA9OPRM1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035406-A4 NOVEL SUBSTITUTED-1H-QUINAZOLINE-2,4-DIONE DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME KOREA RES INST CHEM TECH (KR) 2009-08-05 EP disclosed
EP-2035406-A1 NOVEL SUBSTITUTED-1H-QUINAZOLINE-2,4-DIONE DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Korea Research Institute of Chemical Technology (KR) 2009-03-18 EP disclosed
WO-2008004716-A1 NOVEL SUBSTITUTED-1H-QUINAZOLINE-2,4-DIONE DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME KOREA RESERACH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2008-01-10 WO disclosed