SCHEMBL4394549

SCHEMBL4394549

CC(=O)Nc1cc(C(=N)NO)ccc1F

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.55
HDAC6 Q9UBN7 4/20 0.55
HDAC8 Q9BY41 2/20 0.49
ALDH1A1 P00352 2/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC2 Q92769 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
EP300 Q09472 1/20 0.38
CREBBP Q92793 1/20 0.38
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 2/20 0.37
MAPK1 P28482 1/20 0.37
HTR1F P30939 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4399591 0.84 HDAC6 (0.77) HDAC1HDAC6HDAC8HDAC3KMT2A
SCHEMBL4397000 0.83 HDAC1 (0.49) HDAC1HDAC6HDAC8ALDH1A1CA1
SCHEMBL2055287 0.82 HDAC1 (0.54) HDAC1HDAC6HDAC8ALDH1A1CA1
SCHEMBL16234575 0.80 MEN1 (0.54) HDAC1HDAC6HDAC8ALDH1A1CA1
SCHEMBL15047091 0.79 HDAC1 (0.51) HDAC1HDAC6HDAC8ALDH1A1CA1
SCHEMBL4398972 0.79 HDAC1 (0.51) HDAC1HDAC6HDAC8ALDH1A1CA1
SCHEMBL4395273 0.78 HDAC1 (0.48) HDAC1HDAC6HDAC8NPC1RAB9A
SCHEMBL3276320 0.77 HDAC1 (0.47) HDAC1HDAC6HDAC8ALDH1A1CA1
SCHEMBL2486357 0.76 HDAC1 (0.49) HDAC1HDAC6HDAC8ALDH1A1CA1
SCHEMBL2486361 0.76 HDAC1 (0.49) HDAC1HDAC6HDAC8ALDH1A1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed