SCHEMBL4399591

SCHEMBL4399591

CC(=O)Nc1cc(C(=O)NO)ccc1F

nearest known ligand 0.77

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 18/20 0.77
HDAC1 Q13547 16/20 0.77
HDAC8 Q9BY41 11/20 0.68
ACLY P53396 1/20 0.47
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC11 Q96DB2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2055287 0.84 HDAC1 (0.54) HDAC6HDAC1HDAC8MEN1KMT2A
SCHEMBL4394549 0.84 HDAC1 (0.55) HDAC6HDAC1HDAC8MEN1KMT2A
SCHEMBL16234575 0.83 MEN1 (0.54) HDAC6HDAC1HDAC8ACLYMEN1
SCHEMBL4398972 0.81 HDAC1 (0.51) HDAC6HDAC1HDAC8ACLYKMT2A
SCHEMBL15047091 0.81 HDAC1 (0.51) HDAC6HDAC1HDAC8MEN1KMT2A
SCHEMBL4397000 0.79 HDAC1 (0.49) HDAC6HDAC1HDAC8HDAC3
SCHEMBL2486357 0.79 HDAC1 (0.49) HDAC6HDAC1HDAC8MEN1KMT2A
SCHEMBL2486361 0.79 HDAC1 (0.49) HDAC6HDAC1HDAC8MEN1KMT2A
SCHEMBL4796769 0.77 ALDH1A1 (0.54) HDAC6HDAC1MEN1KMT2A
SCHEMBL30748254 0.77 SMN1; SMN2 (0.55) HDAC6HDAC1MEN1KMT2AHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed