SCHEMBL4397000

SCHEMBL4397000

CC(=O)Nc1cc(C(=N)N)ccc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.49
HDAC6 Q9UBN7 2/20 0.49
KLK1 P06870 3/20 0.46
KLK5 Q9Y337 2/20 0.46
F10 P00742 2/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
PLAU P00749 4/20 0.44
HDAC8 Q9BY41 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC2 Q92769 1/20 0.43
NCOR2 Q9Y618 1/20 0.43
NEU3 Q9UQ49 1/20 0.42
PRSS1 P07477 4/20 0.42
F2 P00734 3/20 0.42
PRSS2 P07478 2/20 0.42
PRSS3 P35030 2/20 0.42
TMPRSS6 Q8IU80 1/20 0.42
ST14 Q9Y5Y6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7902823 0.87 HDAC1 (0.65) HDAC1HDAC6KLK1KLK5F10
SCHEMBL4398972 0.87 HDAC1 (0.51) HDAC1HDAC6F10CA1CA2
SCHEMBL2055287 0.83 HDAC1 (0.54) HDAC1HDAC6CA1CA2CA9
SCHEMBL4394549 0.83 HDAC1 (0.55) HDAC1HDAC6CA1CA2CA9
SCHEMBL16234575 0.81 MEN1 (0.54) HDAC1HDAC6CA1CA2CA9
SCHEMBL15047091 0.80 HDAC1 (0.51) HDAC1HDAC6CA1CA2CA9
SCHEMBL7903346 0.79 KLK1 (0.56) HDAC1HDAC6KLK1KLK5F10
SCHEMBL4399591 0.79 HDAC6 (0.77) HDAC1HDAC6HDAC8HDAC3
SCHEMBL7894917 0.77 CA1 (0.55) HDAC1HDAC6F10CA1CA2
SCHEMBL2486357 0.77 HDAC1 (0.49) HDAC1HDAC6CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed