SCHEMBL4395036

SCHEMBL4395036

N=C(NO)c1ccc2[nH]c(=O)[nH]c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.44
MAPT P10636 6/20 0.42
KDM4E B2RXH2 4/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
LMNA P02545 1/20 0.42
MAPK1 P28482 1/20 0.41
GAA P10253 2/20 0.41
BCL6 P41182 3/20 0.40
BCOR Q6W2J9 3/20 0.40
POLB P06746 1/20 0.40
ALDH1A1 P00352 5/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
PKM P14618 1/20 0.40
THRB P10828 1/20 0.39
KLK7 P49862 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDE3B Q13370 2/20 0.39
PDE3A Q14432 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4399623 0.84 SMYD3 (0.47) SMYD3MAPTKDM4EMEN1KMT2A
SCHEMBL1829208 0.76 RXFP1 (0.50) SMYD3MAPTKDM4EKMT2AGAA
SCHEMBL12348283 0.76 KIF11 (0.40) MAPTKDM4EMEN1KMT2AGAA
SCHEMBL1423203 0.73 NOS1 (0.50) SMYD3KDM4EMEN1KMT2ALMNA
SCHEMBL1095502 0.73 SIRT2 (0.69) SMYD3MAPTKDM4EMEN1KMT2A
SCHEMBL4422966 0.72 BCL6 (0.60) SMYD3MAPTKDM4EMEN1KMT2A
SCHEMBL1119917 0.72 MAPT (0.57) SMYD3MAPTKDM4EMEN1KMT2A
SCHEMBL29511878 0.72 BCL6 (0.60) SMYD3MAPTKDM4EMEN1KMT2A
SCHEMBL28431190 0.72 MAPT (0.49) SMYD3MAPTKDM4EMEN1KMT2A
SCHEMBL474689 0.71 BCL6 (0.64) MAPTKDM4EMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed