SCHEMBL4396249

SCHEMBL4396249

NCc1cccc(C2CCN(C(=O)c3cc4scc(Cl)c4s3)CC2)c1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 12/20 0.48
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
KCNH2 Q12809 1/20 0.47
F10 P00742 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4411514 0.94 TPSAB1 (0.56) TPSAB1F10
SCHEMBL4395877 0.79 TPSAB1 (0.55) TPSAB1CYP3A4CYP2D6KCNH2
Trifluoroacetic Acid SCHEMBL4410369 0.79 TPSAB1 (0.57) TPSAB1F10
SCHEMBL15772184 0.77 CYP3A4 (0.53) TPSAB1CYP3A4CYP2D6KCNH2
SCHEMBL15780781 0.76 TPSAB1 (0.54) TPSAB1CYP3A4CYP2D6KCNH2
Trifluoroacetic Acid SCHEMBL4395571 0.76 TPSAB1 (0.59) TPSAB1F10
Hydrochloric Acid SCHEMBL4408023 0.75 TPSAB1 (0.53) TPSAB1CYP3A4CYP2D6KCNH2
SCHEMBL4411520 0.75 TPSAB1 (0.55) TPSAB1
Trifluoroacetic Acid SCHEMBL4398774 0.75 TPSAB1 (0.59) TPSAB1F10
Trifluoroacetic Acid SCHEMBL4409332 0.75 TPSAB1 (0.55) TPSAB1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296972-B1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS AVENTIS PHARMA INC (US) 2009-12-23 EP claimed
US-6977263-B2 Chemical compounds AVENTIS PHARMACEUTICALS INC. (US) 2005-12-20 US disclosed