SCHEMBL4397754

SCHEMBL4397754

N=C(NO)c1ccnc(N2CCSCC2)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.43
BRAF P15056 1/20 0.40
MAPK13 O15264 1/20 0.34
PROKR1 Q8TCW9 4/20 0.34
ALDH1A1 P00352 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPK10 P53779 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CNR2 P34972 1/20 0.33
HRH3 Q9Y5N1 2/20 0.33
CTSA P10619 1/20 0.33
ACHE P22303 2/20 0.33
JAK2 O60674 1/20 0.32
FLT3 P36888 1/20 0.32
PRMT5 O14744 1/20 0.32
PRKDC P78527 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4398938 0.85 HRH4 (0.46) PIK3CAPROKR1ALDH1A1CTSAPRMT5
SCHEMBL4411361 0.83 PIK3CA (0.63) PIK3CABRAFMAPK13ALDH1A1PRMT5
SCHEMBL1791657 0.78 PIK3CA (0.68) PIK3CABRAFALDH1A1
SCHEMBL15450883 0.73 GRIN2D (0.53) ALDH1A1ALOX15MAPK10HSD17B10
SCHEMBL28978587 0.70 GRIN2D (0.53) ALDH1A1ALOX15MAPK10HSD17B10
SCHEMBL4392713 0.70 LOXL2 (0.49) ALDH1A1ALOX15HSD17B10
SCHEMBL4409309 0.70 PRMT5 (0.43) ALDH1A1MAPK10PRMT5
SCHEMBL4394180 0.68 KDM4D (0.31) ALDH1A1
SCHEMBL2134993 0.68 KDM1A (0.42) ALDH1A1
SCHEMBL12651287 0.67 POLB (0.44) PIK3CAALDH1A1ALOX15MAPK10HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed