SCHEMBL4399808

SCHEMBL4399808

COC(=O)C(CNc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.51
CTSK P43235 6/20 0.48
CTSS P25774 5/20 0.48
CTSL P07711 1/20 0.48
CTSB P07858 1/20 0.48
PPARA Q07869 5/20 0.47
PPARG P37231 4/20 0.47
ATM Q13315 1/20 0.47
NFKB1 P19838 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
ACE P12821 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
PPARD Q03181 2/20 0.46
HDAC8 Q9BY41 1/20 0.45
SYK P43405 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13258281 0.82 ATM (0.50) CTSKCTSSCTSLCTSBPPARA
SCHEMBL13257955 0.82 ATM (0.50) CTSKCTSSCTSLCTSBPPARA
SCHEMBL13257888 0.82 ATM (0.50) CTSKCTSSCTSLCTSBPPARA
SCHEMBL203084 0.82 ATM (0.67) KLK5CTSKCTSSCTSLCTSB
SCHEMBL29901268 0.82 ATM (0.67) KLK5CTSKCTSSCTSLCTSB
SCHEMBL9977267 0.82 ATM (0.67) KLK5CTSKCTSSCTSLCTSB
SCHEMBL3866896 0.82 PPARA (0.49) KLK5CTSKCTSSCTSLCTSB
SCHEMBL6292728 0.81 KLK5 (0.72) KLK5CTSKCTSSCTSLCTSB
SCHEMBL21473748 0.81 KLK5 (0.72) KLK5CTSKCTSSCTSLCTSB
SCHEMBL84524 0.81 KLK5 (0.72) KLK5CTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2233483-B1 Indole or Benzimidazole derivatives as IkB-kinase modulators and intermediates in their preparation. SANOFI AVENTIS DEUTSCHLAND (DE) 2012-05-09 EP disclosed