SCHEMBL4400941

SCHEMBL4400941

Cc1ccc(C(=O)c2ccc(C)nc2)cn1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.64
HDAC6 Q9UBN7 1/20 0.64
KDM4E B2RXH2 2/20 0.51
LMNA P02545 2/20 0.48
ALDH1A1 P00352 1/20 0.48
KMT2A Q03164 3/20 0.46
RXFP1 Q9HBX9 2/20 0.44
NPC1 O15118 2/20 0.44
KCNQ3 O43525 1/20 0.44
KCNQ2 O43526 1/20 0.44
MAPT P10636 1/20 0.44
PRKAB2 O43741 1/20 0.43
PRKAG1 P54619 1/20 0.43
PRKAA2 P54646 1/20 0.43
PRKAA1 Q13131 1/20 0.43
PRKAG3 Q9UGI9 1/20 0.43
PRKAG2 Q9UGJ0 1/20 0.43
PRKAB1 Q9Y478 1/20 0.43
POLB P06746 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24307418 0.92 ALDH1A1 (0.64) HDAC1HDAC6KDM4ELMNAALDH1A1
SCHEMBL12921446 0.90 HDAC1 (0.55) HDAC1HDAC6KDM4ELMNAALDH1A1
SCHEMBL1773529 0.88 HDAC1 (0.58) HDAC1HDAC6KDM4ELMNAALDH1A1
SCHEMBL20198329 0.87 ALDH1A1 (0.53) HDAC1HDAC6LMNAALDH1A1KMT2A
SCHEMBL30544993 0.84 HDAC1 (0.62) HDAC1HDAC6KDM4EALDH1A1MAPT
SCHEMBL31290288 0.84 HDAC1 (0.62) HDAC1HDAC6KDM4ELMNAALDH1A1
SCHEMBL575041 0.84 HDAC1 (0.62) HDAC1HDAC6KDM4ELMNAALDH1A1
SCHEMBL181465 0.84 HDAC1 (0.62) HDAC1HDAC6KDM4EALDH1A1MAPT
SCHEMBL4033393 0.84 CCR9 (0.57) HDAC1HDAC6KDM4EALDH1A1KMT2A
SCHEMBL600144 0.82 HDAC1 (0.60) HDAC1HDAC6KDM4ELMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103664754-A New method for preparing 1-(6-methylpyridine-3-yl)-2-[4-(methylsulfanyl)phenyl]acetone UNIV SHANGHAI JIAOTONG 2014-03-26 CN claimed
EP-1675930-B1 NEW MATERIALS FOR ELECTROLUMINESCENCE AND THE UTILIZATION THEREOF MERCK PATENT GMBH (DE) 2018-05-30 EP disclosed
CN-103664754-B Prepare 1-(6-picoline-3-yl)-2-[4-methyl mercapto-phenyl] method of ethyl ketone SHANGHAI JIAO TONG UNIVERSITY (CN) 2016-05-25 CN disclosed
CN-104086565-A FUSED, SPIROCYCLIC HETEROAROMATIC COMPOUNDS FOR THE TREATMENT OF BACTERIAL INFECTIONS ASTRAZENECA AB 2014-10-08 CN disclosed
CN-102171204-B 8-substituted isoquinoline derivative and application thereof ASAHI KASEI PHARMA CORP 2014-08-20 CN disclosed
CN-103664754-A New method for preparing 1-(6-methylpyridine-3-yl)-2-[4-(methylsulfanyl)phenyl]acetone UNIV SHANGHAI JIAOTONG 2014-03-26 CN disclosed
CN-102625799-A Heterocyclic compounds and their uses AMGEN INC 2012-08-01 CN disclosed
US-8173276-B2 Materials for electroluminescence and the utilization thereof MERCK PATENT GMBH (DE) 2012-05-08 US disclosed
US-8173276-B2 Materials for electroluminescence and the utilization thereof MERCK PATENT GMBH (DE) 2012-05-08 US disclosed
CN-102245605-A Fused, spirocyclic heteroaromatic compounds for the treatment of bacterial infections ASTRAZENECA AB 2011-11-16 CN disclosed
CN-102171204-A 8-substituted isoquinoline derivative and application thereof ASAHI KASEI PHARMA CORP 2011-08-31 CN disclosed
CN-102066337-A 5-hydroxypyrimidine-4-carboxamide compounds DAIICHI SANKYO CO LTD 2011-05-18 CN disclosed
US-20100102305-A1 MATERIALS FOR ELECTROLUMINESCENCE AND THE UTILIZATION THEREOF MERCK PATENT GMBH (DE) 2010-04-29 US disclosed
US-20100102305-A1 MATERIALS FOR ELECTROLUMINESCENCE AND THE UTILIZATION THEREOF MERCK PATENT GMBH (DE) 2010-04-29 US disclosed
US-7659540-B2 Materials for electroluminescence and the utilization thereof MERCK PATENT GMBH (DE) 2010-02-09 US disclosed
US-7659540-B2 Materials for electroluminescence and the utilization thereof MERCK PATENT GMBH (DE) 2010-02-09 US disclosed
US-20070080343-A1 New materials for electroluminescence and the utilization thereof MERCK PATENT GMBH (DE) 2007-04-12 US disclosed
US-20070080343-A1 New materials for electroluminescence and the utilization thereof MERCK PATENT GMBH (DE) 2007-04-12 US disclosed