SCHEMBL4401152

SCHEMBL4401152

N=C(NO)c1cccc(N2CCCS2(=O)=O)c1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.61
TP53 P04637 8/20 0.57
MAPT P10636 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.49
SLC9A3 P48764 1/20 0.39
CDK1 P06493 4/20 0.39
CDK4 P11802 4/20 0.39
CDK2 P24941 4/20 0.39
CTSD P07339 1/20 0.38
BACE1 P56817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18929761 0.83 CA1 (0.46) POLBTP53MAPT
SCHEMBL4397150 0.80 POLB (0.91) POLBTP53MAPTSMN1; SMN2CTSD
SCHEMBL6828696 0.80 TP53 (0.67) POLBTP53MAPTSMN1; SMN2
SCHEMBL14584575 0.79 POLB (0.70) POLBTP53MAPTSMN1; SMN2CTSD
SCHEMBL1787817 0.75 POLB (0.56) POLBTP53MAPTSMN1; SMN2SLC9A3
SCHEMBL2187675 0.75 POLB (0.60) POLBTP53MAPTSMN1; SMN2SLC9A3
SCHEMBL4833669 0.74 TP53 (0.64) POLBTP53MAPTSMN1; SMN2
SCHEMBL13745531 0.72 POLB (0.56) POLBTP53MAPTSMN1; SMN2SLC9A3
SCHEMBL12547064 0.72 POLB (0.56) POLBTP53MAPTSMN1; SMN2SLC9A3
SCHEMBL10192187 0.72 TP53 (0.64) POLBTP53MAPTSMN1; SMN2SLC9A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed